SCHEMBL30211016

SCHEMBL30211016

NS(=O)(=O)c1cccc(-c2ccc(OC(F)(F)F)cc2)c1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.51
TRPV1 Q8NER1 2/20 0.45
PTGS2 P35354 2/20 0.43
PTGS1 P23219 1/20 0.43
PTGES2 Q9H7Z7 3/20 0.43
SCN10A Q9Y5Y9 1/20 0.43
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
KIF11 P52732 1/20 0.40
KIT P10721 1/20 0.40
KDR P35968 1/20 0.40
FLT3 P36888 1/20 0.40
ABL1 P00519 3/20 0.38
BCR P11274 2/20 0.38
F10 P00742 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30211043 0.85 SCN9A (0.60) SCN9ATRPV1PTGS2PTGS1PTGES2
SCHEMBL1069769 0.82 PTGES2 (0.42) SCN9APTGS2PTGS1PTGES2CA1
SCHEMBL27702233 0.75 CA2 (0.47) PTGES2CA1CA2KIF11
SCHEMBL8631562 0.75 TRPV1 (0.50) SCN9ATRPV1PTGS2PTGS1PTGES2
SCHEMBL14572634 0.74 SCN9A (0.47) SCN9ATRPV1PTGS2PTGS1SCN10A
SCHEMBL8631700 0.71 TRPV1 (0.47) SCN9ATRPV1PTGS2CA1CA2
SCHEMBL17840231 0.71 GPR3 (0.50) KIF11ABL1BCR
SCHEMBL18118195 0.71 PTGS2 (0.68) PTGS2PTGS1CA1CA2KIF11
SCHEMBL5518064 0.70 SLC6A4 (0.55) SCN9APTGES2SCN10ACA1CA2
SCHEMBL12952695 0.70 KIF11 (0.40) SCN9ATRPV1PTGS2PTGS1KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4367103-A1 INHIBITORS OF ALPHA-HEMOLYSIN OF STAPHYLOCOCCUS AUREUS Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2024-05-15 EP disclosed
WO-2023280970-A1 INHIBITORS OF ALPHA-HEMOLYSIN OF STAPHYLOCOCCUS AUREUS Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2023-01-12 WO disclosed