SCHEMBL30258024

SCHEMBL30258024

COCCn1cnc2cc(Br)cc(C(=O)OC)c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPK1 P28482 2/20 0.38
PDE4A P27815 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
TSHR P16473 3/20 0.36
LMNA P02545 2/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PTGER4 P35408 1/20 0.35
OPRK1 P41145 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
HPGD P15428 1/20 0.34
NR3C1 P04150 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25262955 1.00 ACHE (0.44) ACHEMEN1KMT2AMAPK1PDE4A
SCHEMBL25395444 0.80 TSHR (0.34) ACHEMAPK1TSHRLMNAUSP2
SCHEMBL29495175 0.80 TSHR (0.34) ACHEMAPK1TSHRLMNAUSP2
SCHEMBL25259206 0.78 ACHE (0.40) ACHEMEN1KMT2AMAPK1TSHR
SCHEMBL30198194 0.78 ACHE (0.40) ACHEMEN1KMT2AMAPK1TSHR
SCHEMBL25374507 0.75 KDM4E (0.46) USP2ALDH1A1SMN1; SMN2NR3C1
SCHEMBL30552955 0.75 KDM4E (0.46) USP2ALDH1A1SMN1; SMN2NR3C1
SCHEMBL15054540 0.74 LMNA (0.44) MEN1KMT2AMAPK1TSHRLMNA
SCHEMBL31698506 0.74 MEN1 (0.45) ACHEMEN1KMT2APDE4AADORA2A
SCHEMBL23925485 0.73 OPRK1 (0.43) ALDH1A1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115443268-A Benzimidazole derivatives 豪夫迈·罗氏有限公司 2022-12-06 CN disclosed