SCHEMBL302933

SCHEMBL302933

O=C1COc2ccc(Cl)cc2N1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.65
PARP1 P09874 3/20 0.59
MAPT P10636 6/20 0.57
ALDH1A1 P00352 4/20 0.57
KMT2A Q03164 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
DRD4 P21917 1/20 0.55
THRB P10828 1/20 0.53
KDM4E B2RXH2 1/20 0.52
CMA1 P23946 1/20 0.51
AHR P35869 1/20 0.51
PKM P14618 1/20 0.51
POLB P06746 1/20 0.51
NR3C2 P08235 2/20 0.50
TRPV1 Q8NER1 1/20 0.50
NR3C1 P04150 1/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30015279 1.00 MMP12 (0.65) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL5987554 0.98 MMP12 (0.63) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL304249 0.86 DRD4 (0.56) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL15964651 0.83 AHR (0.49) MMP12PARP1MAPTDRD4CMA1
SCHEMBL8490860 0.80 MMP12 (0.41) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL6321386 0.80 NR3C2 (0.58) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL279594 0.79 MMP12 (1.00) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL861110 0.79 MMP12 (0.65) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL277585 0.79 MMP12 (0.65) MMP12PARP1MAPTALDH1A1KMT2A
SCHEMBL707058 0.79 MMP12 (0.65) MMP12PARP1ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 131 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084815-A Synthesis method of 7-bromo-6-chloro-3, 4-dihydro-2H-1, 4-benzoxazine 南通大学 2024-05-28 CN claimed
WO-2025099111-A1 NEW TELESCOPING SYNTHESES OF 6-HYDROXY-BENZOMORPHOLINE (3,4-DIHYDRO-2H-1,4-BENZOXAZIN-6-OL) WELLA GERMANY GMBH (DE) 2025-05-15 WO disclosed
CN-118084815-A Synthesis method of 7-bromo-6-chloro-3, 4-dihydro-2H-1, 4-benzoxazine 南通大学 2024-05-28 CN disclosed
CN-110092782-B Benzo-hexaazacyclo compound and preparation method and application thereof 中国科学院广州生物医药与健康研究院 2022-10-21 CN disclosed
US-20210380570-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. 2021-12-09 US disclosed
EP-3790551-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2021-03-17 EP disclosed
US-10851215-B2 Graphene-augmented composite materials THE BOEING COMPANY (US) 2020-12-01 US disclosed
WO-2019217307-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2019-11-14 WO disclosed
WO-2019217307-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2019-11-14 WO disclosed
US-20190338087-A1 GRAPHENE-AUGMENTED COMPOSITE MATERIALS THE BOEING COMPANY (US) 2019-11-07 US disclosed
US-20060173183-A1 Multicyclic bis-amide MMP inhibitors ALANTOS PHARMACEUTICALS, INC., 2006-08-03 US disclosed
EP-1660431-A2 PHENOXYACETIC ACID DERIVATIVES Astrazeneca AB (SE) 2006-05-31 EP disclosed
US-20050222148-A1 Phenylaminopropanol derivatives and methods of their use WYETH (US) 2005-10-06 US disclosed
US-20050222142-A1 Phenylaminopropanol derivatives and methods of their use WYETH (US) 2005-10-06 US disclosed
WO-2005018529-A2 PHENOXIACETIC ACID DERIVATIVES ASTRAZENECA AB (SE) 2005-03-03 WO disclosed
EP-0769495-B1 Fungicides ZENECA LTD (GB) 1999-04-21 EP disclosed
US-5830890-A NITROGEN HETEROCYCLE ATTACHED THROUGH OXYMETHYLENE GROUP TO PHENYL RING WITH O-METHYL 3-METHOXYACRYLATE OR WITH METHYL 3-METHOXYIMINOACETATE OR AMIDE DERIVATIVE ZENECA LIMITED (GB) 1998-11-03 US disclosed
EP-0858997-A1 Fungicides ZENECA LIMITED (GB) 1998-08-19 EP disclosed
EP-0769495-A1 Fungicides ZENECA LIMITED (GB) 1997-04-23 EP disclosed
US-3935203-A ANALGESICS, ANTI-OEDEMATOUS CERPHA (FR) 1976-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050222148-A1 Phenylaminopropanol derivatives and methods of their use PAH, PNMT, COMT MMP12 2805/4885PARP1 1187/4885MAPT 2326/4885
US-20210380570-A1 KRAS G12C INHIBITORS KRAS, NRAS, HRAS MMP12 1433/4885PARP1 1128/4885MAPT 3928/4885
US-20060173183-A1 Multicyclic bis-amide MMP inhibitors MMP13, MMP3, MMP11 MMP12 7/4885PARP1 190/4885MAPT 2159/4885
US-20050222142-A1 Phenylaminopropanol derivatives and methods of their use PAH, PNMT, COMT MMP12 2805/4885PARP1 1187/4885MAPT 2326/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.