SCHEMBL30306325

SCHEMBL30306325

c1ccc(COCCCOc2ccccc2N2CCOCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A4 P31645 1/20 0.52
SLC6A3 Q01959 1/20 0.52
ALDH1A1 P00352 4/20 0.48
MAPT P10636 2/20 0.48
GAA P10253 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
POLB P06746 1/20 0.47
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
DRD4 P21917 2/20 0.45
DRD1 P21728 1/20 0.45
DRD5 P21918 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CCR5 P51681 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30306336 0.87 CCR5 (0.55) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL29135294 0.87 CCR5 (0.55) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL30306324 0.83 ALDH1A1 (0.50) ALDH1A1MAPTCNR1CNR2DRD4
SCHEMBL30306331 0.82 DRD2 (0.52) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL29135260 0.82 DRD2 (0.52) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL3921372 0.81 ALDH1A3 (0.49) ALDH1A1MAPTGAANPC1RAB9A
SCHEMBL29135246 0.80 PIK3CG (0.41) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL31008257 0.80 PIK3CG (0.41) HTR1ASLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8342129 0.77 POLB (0.54) ALDH1A1MAPTGAANPC1RAB9A
SCHEMBL29135256 0.77 TSHR (0.46) ALDH1A1GAACNR1CNR2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117957232-A Azaindazole macrocyclic compounds and uses thereof 北京伯汇生物技术有限公司 2024-04-30 CN disclosed
CN-115838373-A Azaindazole macrocycles and uses thereof 北京伯汇生物技术有限公司 2023-03-24 CN disclosed