SCHEMBL29135260

SCHEMBL29135260

CN1CCN(c2ccccc2OCCCCOCc2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.52
DRD3 P35462 3/20 0.52
HTR1A P08908 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A4 P31645 1/20 0.52
SLC6A3 Q01959 1/20 0.52
DRD4 P21917 1/20 0.50
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
ADRA1D P25100 1/20 0.47
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
AVPR2 P30518 6/20 0.47
AVPR1A P37288 6/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30306331 1.00 DRD2 (0.52) DRD2DRD3HTR1ASLC6A2SLC6A4
SCHEMBL14355885 0.86 HTR1A (0.68) DRD2DRD3HTR1ASLC6A2SLC6A4
SCHEMBL30306319 0.86 HSP90AB1 (0.41) DRD2DRD3
SCHEMBL29135242 0.86 HSP90AB1 (0.41) DRD2DRD3
SCHEMBL30306325 0.82 HTR1A (0.52) DRD2DRD3HTR1ASLC6A2SLC6A4
SCHEMBL9332845 0.80 DRD2 (0.67) DRD2DRD3HTR1ADRD4ALDH1A1
SCHEMBL8720341 0.80 ADRA1D (0.65) DRD2DRD3HTR1AKDM4EALDH1A1
SCHEMBL30306326 0.80 HRH4 (0.49) KDM4EALDH1A1TDP1
SCHEMBL24712696 0.80 DRD2 (0.56) DRD2DRD3HTR1AKDM4EALDH1A1
SCHEMBL8894896 0.79 ALDH1A1 (0.57) DRD2DRD3HTR1AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117957232-A Azaindazole macrocyclic compounds and uses thereof 北京伯汇生物技术有限公司 2024-04-30 CN disclosed
CN-115838373-A Azaindazole macrocycles and uses thereof 北京伯汇生物技术有限公司 2023-03-24 CN disclosed