SCHEMBL30367171

SCHEMBL30367171

COc1cc(N(C)c2cc(C)nc3ccccc23)cc(OC)c1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.48
RAD52 P43351 1/20 0.48
LMNA P02545 3/20 0.46
GAA P10253 2/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
KDM1A O60341 1/20 0.45
EGFR P00533 3/20 0.45
GAK O14976 1/20 0.45
RIPK2 O43353 1/20 0.45
STK16 O75716 1/20 0.45
AAK1 Q2M2I8 1/20 0.45
BMP2K Q9NSY1 1/20 0.45
NLK Q9UBE8 1/20 0.45
IRAK3 Q9Y616 1/20 0.45
NPC1 O15118 1/20 0.44
PDGFRB P09619 3/20 0.43
PDGFRA P16234 1/20 0.43
KDR P35968 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30366693 0.87 LMNA (0.49) LMNAGAATP53TSHRSMN1; SMN2
SCHEMBL21882934 0.81 NCF1 (0.48) POLBLMNAGAATP53TSHR
SCHEMBL6592363 0.81 SMN1; SMN2 (0.46) POLBRAD52LMNAGAATP53
SCHEMBL2257287 0.79 PDGFRB (0.70) POLBRAD52EGFRPDGFRBPDGFRA
SCHEMBL30367104 0.77 CYP1A2 (0.50) KDM1AEGFRPDGFRBKDRCYP1A2
SCHEMBL30367038 0.77 CYP1A2 (0.50) LMNATP53TSHRSMN1; SMN2KDM1A
SCHEMBL30367213 0.76 CYP1A2 (0.49) LMNATSHRSMN1; SMN2KDM1AEGFR
SCHEMBL6790532 0.73 CYP1A2 (0.60) KDM1ACYP1A2
SCHEMBL266444 0.73 LMNA (0.64) POLBLMNAGAATP53TSHR
SCHEMBL29877118 0.73 LMNA (0.64) POLBLMNAGAATP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825610-B 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-03-31 CN disclosed