SCHEMBL303909

SCHEMBL303909

COC(=O)c1ccc2c(c1)OCC(=O)N2

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
LMNA P02545 2/20 0.52
MAPT P10636 4/20 0.50
ALOX5 P09917 1/20 0.50
POLB P06746 1/20 0.50
GAA P10253 2/20 0.49
CRBN Q96SW2 1/20 0.48
PKM P14618 1/20 0.47
PARP1 P09874 1/20 0.47
NSD2 O96028 2/20 0.47
MMP12 P39900 1/20 0.47
CYP3A4 P08684 1/20 0.46
CYP19A1 P11511 1/20 0.46
CYP2C9 P11712 1/20 0.46
TRPV1 Q8NER1 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978611 1.00 ALDH1A1 (0.52) ALDH1A1LMNAMAPTALOX5POLB
SCHEMBL6752 0.89 ALDH1A1 (0.63) ALDH1A1LMNAMAPTALOX5POLB
SCHEMBL29901720 0.89 ALDH1A1 (0.63) ALDH1A1LMNAMAPTALOX5POLB
SCHEMBL7349545 0.84 ALDH1A1 (0.52) ALDH1A1LMNAMAPTPOLBGAA
SCHEMBL23611043 0.83 ALOX5 (0.48) ALDH1A1LMNAMAPTALOX5CRBN
SCHEMBL25720031 0.82 GAA (0.52) ALDH1A1MAPTPOLBGAAPKM
SCHEMBL941445 0.82 GAA (0.56) ALDH1A1LMNAMAPTALOX5GAA
SCHEMBL13932092 0.81 ALDH1A1 (0.57) ALDH1A1LMNAMAPTPOLBGAA
SCHEMBL4265304 0.81 ALDH1A1 (0.57) ALDH1A1LMNAMAPTPOLBGAA
SCHEMBL3283784 0.81 ALDH1A1 (0.56) ALDH1A1LMNAMAPTPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 85 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12637426-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors MISSION THERAPEUTICS LIMITED (GB) 2026-05-26 US disclosed
EP-4384268-B1 SMALL MOLECULE UREA DERIVATIVES AS STING ANTAGONISTS CURADEV PHARMA PVT LTD (IN) 2026-03-18 EP disclosed
US-20250074904-A1 NSD2-TARGETED CHECMICAL DEGRADERTS AND COMPOSITIONS AND METHODS OF USE THEREOF THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2025-03-06 US disclosed
CN-115151304-B Small molecule interferon gene stimulating factor (STING) antagonists 库拉德夫制药私人有限公司 2025-02-11 CN disclosed
US-20240360119-A1 SMALL MOLECULE UREA DERIVATIVES AS STING ANTAGONISTS CURADEV PHARMA PVT. LTD. (IN) 2024-10-31 US disclosed
EP-4384268-A1 SMALL MOLECULE UREA DERIVATIVES AS STING ANTAGONISTS Curadev Pharma Pvt. Ltd. (IN) 2024-06-19 EP disclosed
CN-118019738-A Small molecule urea derivatives as STING antagonists 库拉德夫制药私人有限公司 2024-05-10 CN disclosed
WO-2023091565-A1 NSD2-TARGETED CHEMICAL DEGRADERS AND COMPOSITIONS AND METHODS OF USE THEREOF THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2023-05-25 WO disclosed
US-20230124361-A1 SMALL MOLECULE STING ANTAGONISTS CURADEV PHARMA PVT. LTD. (IN) 2023-04-20 US disclosed
US-20230124361-A1 SMALL MOLECULE STING ANTAGONISTS CURADEV PHARMA PVT. LTD. (IN) 2023-04-20 US disclosed
CN-1060769-C 1,4-benzoxazine derivatives, pharmaceutical composition containing the same and use thereof KENEBO LTD (JP) 2001-01-17 CN disclosed
EP-0719766-B1 1,4-Benzoxazine derivative, pharmaceutical composition containing the same and use thereof KANEBO LTD (JP) 2000-04-12 EP disclosed
EP-0543997-B1 DERIVATIVES OF METHOTREXATE WITH ANTIRHEUMATIC ACTIVITY CHUGAI PHARMACEUTICAL CO LTD (JP) 1999-12-08 EP disclosed
US-5597820-A CARDIOVASCULAR DISORDERS KANEBO, LTD. (JP) 1997-01-28 US disclosed
CN-1032858-C Methylamino pterin derivatives CHUGAI PHARMACEUTICAL CO LTD (JP) 1996-09-25 CN disclosed
CN-1130183-A 1,4-benzoxazine derivatives, pharmaceutical composition containing the same and use thereof KANEBO LTD (JP) 1996-09-04 CN disclosed
EP-0719766-A1 1,4-Benzoxazine derivative, pharmaceutical composition containing the same and use thereof KANEBO LTD. (JP) 1996-07-03 EP disclosed
US-5354753-A Methotrexate derivative CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1994-10-11 US disclosed
EP-0543997-A1 NOVEL METHOTREXATE DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 1993-06-02 EP disclosed
CN-1059725-A Novel methotrexate derivatives CHUGAI PHARMACEUTICAL CO LTD (JP) 1992-03-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240360119-A1 SMALL MOLECULE UREA DERIVATIVES AS STING ANTAGONISTS STING1, CGAS, SSB ALDH1A1 3165/4885LMNA 1842/4885MAPT 2509/4885
US-20250074904-A1 NSD2-TARGETED CHECMICAL DEGRADERTS AND COMPOSITIONS AND METHODS OF USE THEREOF NCOR2, NSD2, NCOR1 ALDH1A1 4559/4885LMNA 3179/4885MAPT 2156/4885
US-20230124361-A1 SMALL MOLECULE STING ANTAGONISTS STING1, CGAS, MAVS ALDH1A1 3672/4885LMNA 2127/4885MAPT 3716/4885
US-12637426-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors USP30, USP1, USP10 ALDH1A1 1185/4885LMNA 2783/4885MAPT 2466/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.