SCHEMBL30402499

SCHEMBL30402499

Cc1c(C(=O)NN)cccc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SUCNR1 Q9BXA5 1/20 0.51
PDCD1 Q15116 4/20 0.50
CD274 Q9NZQ7 4/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
MAPT P10636 2/20 0.49
GAA P10253 1/20 0.49
GFER P55789 1/20 0.49
BCAT2 O15382 1/20 0.49
CHRNB2 P17787 2/20 0.47
CHRNB4 P30926 2/20 0.47
CHRNA3 P32297 2/20 0.47
CHRNA4 P43681 2/20 0.47
CTSD P07339 1/20 0.47
RAB9A P51151 1/20 0.47
P2RX7 Q99572 1/20 0.46
HNF4A P41235 1/20 0.46
MYC P01106 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28254835 1.00 SUCNR1 (0.51) SUCNR1PDCD1CD274L3MBTL1MAPT
SCHEMBL29256186 0.85 HDAC7 (0.59) SUCNR1PDCD1CD274L3MBTL1GAA
SCHEMBL6659064 0.84 MKNK1 (0.49) SUCNR1PDCD1CD274L3MBTL1MAPT
SCHEMBL1826396 0.84 CHRNB2 (0.65) MAPTGAAGFERBCAT2CHRNB2
SCHEMBL30345390 0.84 CHRNB2 (0.65) MAPTGAAGFERBCAT2CHRNB2
SCHEMBL28112960 0.83 MYC (0.49) L3MBTL1CTSDRAB9AP2RX7MYC
SCHEMBL7677836 0.83 HNF4A (0.68) L3MBTL1MAPTGAAGFERBCAT2
SCHEMBL436284 0.83 KEAP1 (0.57) SUCNR1PDCD1CD274L3MBTL1CHRNB2
Biphenyl SCHEMBL27596494 0.82 CHRNB2 (0.62) GAABCAT2CHRNB2CHRNB4CHRNA3
SCHEMBL28014189 0.82 L3MBTL1 (0.43) SUCNR1PDCD1CD274L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116041277-B Phenyl and biphenyl substituted five-membered heterocyclic compound, preparation method, pharmaceutical composition and application thereof 中国药科大学 2024-11-01 CN disclosed
CN-115974807-B 2-Phenyl-5-biphenyl-1, 3, 4-oxadiazole compound, preparation method, pharmaceutical composition and application thereof 中国药科大学 2024-05-31 CN disclosed
CN-116041277-A Phenyl and biphenyl substituted five-membered heterocyclic compound, preparation method, pharmaceutical composition and application thereof 中国药科大学 2023-05-02 CN disclosed
CN-115974807-A 2-phenyl-5-biphenyl-1,3,4-oxadiazole compound and preparation method, pharmaceutical composition and application thereof 中国药科大学 2023-04-18 CN disclosed