SCHEMBL30454012

SCHEMBL30454012

Oc1ccc(OCc2ccccc2)nc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.55
LMNA P02545 1/20 0.55
PTGS1 P23219 1/20 0.55
SLC6A2 P23975 1/20 0.55
CYP2C19 P33261 1/20 0.55
PTGS2 P35354 1/20 0.55
SLC6A3 Q01959 1/20 0.55
HIF1A Q16665 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
FFAR1 O14842 1/20 0.49
CXCR2 P25025 1/20 0.47
GABRP O00591 1/20 0.46
GABRD O14764 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL198499 1.00 CYP1A2 (0.55) CYP1A2LMNAPTGS1SLC6A2CYP2C19
Alcohol SCHEMBL29161613 0.93 FFAR1 (0.51) CYP1A2LMNAPTGS1SLC6A2CYP2C19
SCHEMBL1974540 0.84 TSHR (0.44) CYP1A2LMNAPTGS1SLC6A2CYP2C19
SCHEMBL1547117 0.83 LMNA (0.64) CYP1A2LMNAPTGS1SLC6A2CYP2C19
SCHEMBL510464 0.81 FFAR1 (0.47) CYP1A2LMNAPTGS1SLC6A2CYP2C19
Methane SCHEMBL9237648 0.80 CXCR2 (0.44) LMNACXCR2PKMMEN1KMT2A
SCHEMBL510168 0.79 GABRA5 (0.52) LMNAFFAR1CXCR2GABRPGABRD
SCHEMBL16964639 0.79 GABRG2 (0.45) CYP1A2LMNAPTGS1SLC6A2CYP2C19
SCHEMBL12203827 0.79 PKM (0.49) LMNAFFAR1CXCR2GABRPGABRD
SCHEMBL224083 0.79 MAOB (0.56) FFAR1CXCR2GABRPGABRDGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024046221-A1 EGFR INHIBITORS AND USES THEREOF DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2024-03-07 WO disclosed
CN-111787916-B Dihydroceramide desaturase inhibitors for treating diseases 森陶鲁斯治疗公司 2023-09-05 CN disclosed
CN-116669727-A Triazole-pyridinyl substituted azacyclohexylacetic acid compounds as LPA receptor antagonists 唯久生物有限公司 2023-08-29 CN disclosed
EP-4196220-A1 TRIAZOLE-PYRIDINYL SUBSTITUTED AZACYCLOHEXYL ACETIC ACID COMPOUNDS AS LPA RECEPTOR ANTAGONISTS Viva Star Biosciences Limited (HK) 2023-06-21 EP disclosed