SCHEMBL30476366

SCHEMBL30476366

CC(C)(C)OC(=O)N1CCN(Cc2ccc(F)cc2Br)C(=O)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.46
MKNK1 Q9BUB5 1/20 0.42
GPR119 Q8TDV5 2/20 0.41
KDM1A O60341 3/20 0.39
DPP4 P27487 1/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
IDO2 Q6ZQW0 1/20 0.39
ESR2 Q92731 1/20 0.38
NR1H2 P55055 2/20 0.38
PLK1 P53350 1/20 0.38
ALDH1A1 P00352 2/20 0.38
PIK3CD O00329 1/20 0.38
LMNA P02545 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20818471 1.00 P2RX7 (0.46) P2RX7MKNK1GPR119KDM1ADPP4
SCHEMBL20818268 0.89 ALDH1A1 (0.48) P2RX7MKNK1GPR119KDM1ADPP4
SCHEMBL30476344 0.89 ALDH1A1 (0.48) P2RX7MKNK1GPR119KDM1ADPP4
SCHEMBL20818483 0.88 P2RX7 (0.47) P2RX7GPR119KDM1ADPP4IDO1
SCHEMBL30476361 0.88 P2RX7 (0.47) P2RX7GPR119KDM1ADPP4IDO1
SCHEMBL20818026 0.85 P2RX7 (0.45) P2RX7GPR119KDM1ADPP4IDO1
SCHEMBL30476449 0.85 P2RX7 (0.45) P2RX7GPR119KDM1ADPP4IDO1
SCHEMBL25206368 0.85 USP30 (0.45) P2RX7KDM1ADPP4ESR2CYP3A4
SCHEMBL30352468 0.85 USP30 (0.45) P2RX7KDM1ADPP4ESR2CYP3A4
SCHEMBL20818076 0.85 P2RX7 (0.44) P2RX7GPR119KDM1ADPP4PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12435078-B2 Pyridazinones and methods of use thereof GFB (ABC), LLC (US) 2025-10-07 US disclosed
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GFB (ABC), LLC 2023-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF PDXK, ATP6V1B1, REN P2RX7 270/4885MKNK1 1944/4885GPR119 846/4885
US-12435078-B2 Pyridazinones and methods of use thereof PDXK, ATP6V1B1, REN P2RX7 270/4885MKNK1 1944/4885GPR119 846/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.