SCHEMBL30489100

SCHEMBL30489100

OC(c1ccc(Cl)cc1)c1cccnc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.38
HSP90AA1 P07900 3/20 0.37
KDM4E B2RXH2 2/20 0.37
S1PR1 P21453 2/20 0.37
S1PR3 Q99500 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
FFAR2 O15552 1/20 0.37
S1PR4 O95977 1/20 0.37
HPGD P15428 1/20 0.37
KCNA5 P22460 1/20 0.35
KCND3 Q9UK17 1/20 0.35
P4HB P07237 1/20 0.35
PAX8 Q06710 1/20 0.35
PSMD14 O00487 1/20 0.35
MMP2 P08253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707557 1.00 CYP19A1 (0.38) CYP19A1HSP90AA1KDM4ES1PR1S1PR3
SCHEMBL4706109 0.84 SMN1; SMN2 (0.47) KDM4EALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL4182229 0.83 FAAH (0.43) ALDH1A1LMNAMAPTHTTSMN1; SMN2
SCHEMBL4705649 0.83 KCNA5 (0.48) ALDH1A1MAPTSMN1; SMN2L3MBTL1S1PR4
SCHEMBL4707217 0.78 CYP2C19 (0.45) CYP19A1HSP90AA1KDM4ES1PR1ALDH1A1
SCHEMBL14033360 0.78 L3MBTL1 (0.48) HSP90AA1KDM4EALDH1A1LMNAMAPT
SCHEMBL14033102 0.78 HSP90AA1 (0.47) HSP90AA1KDM4ELMNAMAPTHTT
SCHEMBL18322302 0.77 S1PR3 (0.42) CYP19A1S1PR1S1PR3ALDH1A1LMNA
SCHEMBL30489175 0.77 S1PR3 (0.42) CYP19A1S1PR1S1PR3ALDH1A1LMNA
SCHEMBL30251313 0.76 ALDH1A1 (0.40) CYP19A1HSP90AA1S1PR1S1PR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107787322-B Tricyclic compounds and their use as phosphodiesterase inhibitors 辉瑞大药厂 2023-07-07 CN disclosed