SCHEMBL3050301

SCHEMBL3050301

NC1CCc2c(ccc(Cl)c2Cl)C1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.50
DRD3 P35462 5/20 0.50
OPRK1 P41145 1/20 0.47
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR2B P41595 1/20 0.46
PLAU P00749 1/20 0.46
PNMT P11086 2/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11348398 0.82 HTR2A (0.41) DRD2DRD3OPRK1HTR2AHTR2C
Hydrochloric Acid SCHEMBL25287000 0.81 PNMT (0.42) DRD2DRD3HTR2AHTR2CHTR2B
SCHEMBL4263745 0.70 DRD2 (0.64) DRD2DRD3OPRK1PLAUADRA2A
SCHEMBL10618547 0.70 MAPT (0.56) DRD2DRD3OPRK1PLAU
SCHEMBL11578773 0.69 ACHE (0.38) HTR2AHTR2CHTR2BPNMTADRA2A
Bromide SCHEMBL7200937 0.69 DRD2 (0.62) DRD2DRD3OPRK1PLAUADRA2A
SCHEMBL11884613 0.68 MAPT (0.64) DRD2DRD3OPRK1PLAU
SCHEMBL11358755 0.68 ADRA1A (0.34) DRD2DRD3OPRK1PLAUADRA1A
SCHEMBL11359509 0.68 ADRA1A (0.34) DRD2DRD3OPRK1ADRA1A
SCHEMBL24095373 0.68 ADRA1A (0.38) DRD2DRD3OPRK1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100143322-A1 USE OF INHIBITORS OF N-METHYL TRANSFERASES FOR THE THERAPY OF PARKINSON'S DISEASE PLT PATENT & LICENCE TRADING LTD., C/O THE B-NET (GB) 2010-06-10 US claimed
US-20100143322-A1 USE OF INHIBITORS OF N-METHYL TRANSFERASES FOR THE THERAPY OF PARKINSON'S DISEASE PLT PATENT & LICENCE TRADING LTD., C/O THE B-NET (GB) 2010-06-10 US disclosed
US-3919316-A 2-Aminodichlorotetralins LILLY CO ELI 1975-11-11 US disclosed