SCHEMBL30528355

SCHEMBL30528355

CON(C)C(=O)c1cnc(-c2cnccn2)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.39
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 1/20 0.39
CYP1A2 P05177 1/20 0.39
CDC7 O00311 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTT P42858 2/20 0.33
RECQL P46063 1/20 0.33
MAPK8 P45983 1/20 0.33
MAPK9 P45984 1/20 0.33
MAPK10 P53779 1/20 0.33
GRM1 Q13255 1/20 0.33
TERT O14746 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30528397 0.76 PIM2 (0.50) HSD17B10KDM4EALDH1A1CDC7DBF4
SCHEMBL20239488 0.73 TRPM8 (0.40)
SCHEMBL30528350 0.72 GRM1 (0.37) HSD17B10KDM4EALDH1A1HPGDCYP1A2
SCHEMBL2311114 0.71 KDM4E (0.50) HSD17B10KDM4EALDH1A1CYP1A2NPC1
SCHEMBL20239450 0.69 FAAH (0.33)
SCHEMBL10291124 0.67 NPSR1 (0.46) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL17212192 0.66 ALDH1A1 (0.45) KDM4EALDH1A1HPGDCYP1A2NPC1
SCHEMBL21333375 0.66 FAAH (0.43) ALDH1A1NPC1RAB9AMEN1MAPT
SCHEMBL4568047 0.65 CHRNA4 (0.36) TDP1MEN1KMT2A
SCHEMBL434252 0.64 ALDH1A1 (0.59) HSD17B10KDM4EALDH1A1CYP1A2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116600803-A Macrocyclic urea orexin receptor agonists 默沙东有限责任公司 2023-08-15 CN disclosed