SCHEMBL20239488

SCHEMBL20239488

CON(C)C(=O)c1cnc(O)o1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 2/20 0.40
CLK1 P49759 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
MLYCD O95822 1/20 0.33
FAAH O00519 2/20 0.32
OXTR P30559 1/20 0.32
ICAM1 P05362 1/20 0.32
SELE P16581 1/20 0.32
GPR119 Q8TDV5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28869959 0.87 TRPM8 (0.33) TRPM8
SCHEMBL20239450 0.78 FAAH (0.33) CLK1DYRK1ADYRK1BMLYCDFAAH
SCHEMBL21333375 0.74 FAAH (0.43) FAAH
SCHEMBL30528355 0.73 HSD17B10 (0.39)
SCHEMBL10291124 0.72 NPSR1 (0.46)
SCHEMBL4568047 0.70 CHRNA4 (0.36) TRPM8CLK1DYRK1ADYRK1BMLYCD
SCHEMBL20239403 0.69
SCHEMBL4568048 0.68 KLK7 (0.44)
SCHEMBL5269847 0.68 CLK1 (0.33) TRPM8CLK1DYRK1ADYRK1BMLYCD
SCHEMBL6050525 0.68 RAB9A (0.39) CLK1DYRK1ADYRK1BMLYCDFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260055062-A1 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC 2026-02-26 US disclosed
US-12492171-B2 Heterocyclic inhibitors of MCT4 Vettore, LLC (US) 2025-12-09 US disclosed
EP-4442318-A2 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC (US) 2024-10-09 EP disclosed
CN-110114351-B Heterocyclic inhibitors of MCT4 维托尔股份有限公司 2022-09-20 CN disclosed
US-20220251047-A1 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC 2022-08-11 US disclosed
US-11292767-B2 Heterocyclic inhibitors of MCT4 Vettore, LLC (US) 2022-04-05 US disclosed
EP-3551625-A1 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC (US) 2019-10-16 EP disclosed
US-20190112275-A1 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC 2019-04-18 US disclosed
WO-2018111904-A1 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC (US) 2018-06-21 WO disclosed
US-20180162822-A1 HETEROCYCLIC INHIBITORS OF MCT4 Vettore, LLC 2018-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12492171-B2 Heterocyclic inhibitors of MCT4 SLC16A3, SLC16A1, MCTS1 TRPM8 967/4885CLK1 4702/4885DYRK1A 4870/4885
US-11292767-B2 Heterocyclic inhibitors of MCT4 SLC16A3, SLC16A1, MCTS1 TRPM8 967/4885CLK1 4702/4885DYRK1A 4870/4885
US-20190112275-A1 HETEROCYCLIC INHIBITORS OF MCT4 SLC16A3, SLC16A1, MCTS1 TRPM8 967/4885CLK1 4702/4885DYRK1A 4870/4885
US-20220251047-A1 HETEROCYCLIC INHIBITORS OF MCT4 SLC16A3, SLC16A1, MCTS1 TRPM8 967/4885CLK1 4702/4885DYRK1A 4870/4885
US-20180162822-A1 HETEROCYCLIC INHIBITORS OF MCT4 SLC16A3, SLC16A1, MCTS1 TRPM8 967/4885CLK1 4702/4885DYRK1A 4870/4885
US-20260055062-A1 HETEROCYCLIC INHIBITORS OF MCT4 SLC16A1, SLC16A3, SLC16A7 TRPM8 314/4885CLK1 3614/4885DYRK1A 4447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.