SCHEMBL30545928

SCHEMBL30545928

O=C(O)C1CN(C(=O)O)c2cc(F)ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
NOTUM Q6P988 2/20 0.35
ALDH1A1 P00352 2/20 0.34
PDPK1 O15530 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
APEX1 P27695 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
LIPG Q9Y5X9 3/20 0.34
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
STAT1 P42224 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
XIAP P98170 1/20 0.33
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31377997 0.88 NOTUM (0.38) NOTUMALDH1A1LIPGNPC1RAB9A
SCHEMBL31378007 0.77 NOTUM (0.51) NOTUMALDH1A1TDP1MAPT
SCHEMBL31147935 0.72 HDAC2 (0.45) SMN1; SMN2
SCHEMBL28356611 0.72 NOTUM (0.62) KDM4ENOTUMXIAPSLC6A2SLC6A4
SCHEMBL8374944 0.70 LMNA (0.42) KDM4ENOTUMALDH1A1LMNATSHR
SCHEMBL26130366 0.68 BRD4 (0.48) NOTUM
SCHEMBL26130362 0.68 BRD4 (0.48) NOTUM
SCHEMBL5161934 0.67 CHRNB2 (0.40) KDM4EALDH1A1PDPK1LMNAHPGD
SCHEMBL8367941 0.67 MAPT (0.43) NOTUMALDH1A1LMNAHPGDTSHR
SCHEMBL31378019 0.66 CHRM2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114555585-B HPK1 inhibitors and uses thereof 锐格药业公司 2025-02-11 CN disclosed
CN-111944012-B Aromatic amine targeting AR and BET protein degradation chimeric compound and application thereof 海创药业股份有限公司 2023-08-29 CN disclosed