SCHEMBL30549436

SCHEMBL30549436

[2H]C([2H])([2H])NC(=O)c1ccc(NC(=O)NC)nc1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.45
NNMT P40261 1/20 0.44
BAZ2B Q9UIF8 1/20 0.43
EPHX2 P34913 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32677838 0.95 HCAR3 (0.49) HCAR3BAZ2BEPHX2L3MBTL1
SCHEMBL32677808 0.82 HCAR3 (0.42) HCAR3NNMTBAZ2B
SCHEMBL29829392 0.81 NPC1 (0.52) L3MBTL1
SCHEMBL29666324 0.81 NPC1 (0.52) L3MBTL1
SCHEMBL27874609 0.81 HCAR3 (0.69) HCAR3
SCHEMBL28157252 0.80 NNMT (0.70) HCAR3NNMTEPHX2L3MBTL1
SCHEMBL19736133 0.78 PTK2 (0.57) HCAR3NNMTBAZ2B
SCHEMBL31017395 0.77 MAP4K1 (0.47)
SCHEMBL31017468 0.77 MAP4K1 (0.47)
SCHEMBL31017485 0.77 MAP4K1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242546-A1 SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, AND 1,2,4-TRIAZINES AS TYK2 INHIBITORS SUDO BIOSCIENCES LIMITED (GB) 2023-08-03 US claimed
US-20260055121-A1 TYK2 INHIBITORS AND USES THEREOF SUDO BIOSCIENCES LTD (GB) 2026-02-26 US disclosed
CN-117242072-A TYK2 inhibitor and application thereof 苏多生物科学有限公司 2023-12-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242546-A1 SUBSTITUTED PYRIDINES, PYRIDAZINES, PYRIMIDINES, AND 1,2,4-TRIAZINES AS TYK2 INHIBITORS TYK2, PDXK, JAK1 HCAR3 2585/4885NNMT 838/4885BAZ2B 78/4885
US-20260055121-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, CSNK2A3, CSNK2B HCAR3 1546/4885NNMT 1960/4885BAZ2B 484/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.