SCHEMBL30649

SCHEMBL30649

O=C1C=CCC[C@]12Cc1ccc(Br)cc1C2

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.37
CMA1 P23946 1/20 0.36
AHR P35869 1/20 0.36
METAP1 P53582 1/20 0.35
BRD4 O60885 1/20 0.33
PARP10 Q53GL7 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PARP11 Q9NR21 1/20 0.31
PARP1 P09874 1/20 0.31
KDM1A O60341 1/20 0.30
BACE1 P56817 1/20 0.30
PNMT P11086 1/20 0.30
ASIC3 Q9UHC3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30493 0.84 TDP2 (0.39) TDP2CMA1AHRMETAP1BRD4
SCHEMBL9958538 0.76 TDP2 (0.46) TDP2CMA1AHRMETAP1BRD4
SCHEMBL1465537 0.73 TDP1 (0.41) TDP2CMA1AHRMETAP1BRD4
SCHEMBL1464250 0.70 TDP1 (0.39) TDP2CMA1AHRMETAP1BRD4
SCHEMBL11073635 0.69 TDP2 (0.47) TDP2CMA1AHRMETAP1BRD4
SCHEMBL19586472 0.69 TDP2 (0.44) TDP2CMA1AHRMETAP1BRD4
SCHEMBL9958457 0.69 TDP2 (0.41) TDP2CMA1AHRMETAP1BRD4
SCHEMBL9959281 0.69 BACE1 (0.40) TDP2CMA1AHRMETAP1BRD4
SCHEMBL18543791 0.67 TDP2 (0.36) TDP2CMA1AHRMETAP1BRD4
SCHEMBL9958466 0.67 BACE1 (0.40) TDP2CMA1AHRMETAP1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406240-A2 INHIBITORS OF BETA-SECRETASE Vitae Pharmaceuticals, Inc. (US) 2012-01-18 EP disclosed
WO-2010105179-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-09-16 WO disclosed