SCHEMBL30672148

SCHEMBL30672148

Cc1c(Cl)cc(C(N)=O)c(=O)n1-c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MERTK Q12866 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
MARS1 P56192 1/20 0.39
HSD11B1 P28845 1/20 0.38
MAT2A P31153 2/20 0.38
ADRA1D P25100 2/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
PLK4 O00444 1/20 0.38
ROCK2 O75116 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29626186 0.85 POLB (0.44) NPSR1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL30672466 0.82 ALDH1A1 (0.43) NPSR1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL30672493 0.81 ALDH1A1 (0.43) NPSR1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL30672459 0.81 SMN1; SMN2 (0.38) NPSR1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL30672509 0.79 PLAUR (0.36) MERTKNPSR1SMN1; SMN2ALDH1A1KDM4E
SCHEMBL30672116 0.78 BRD4 (0.41) MERTKNPSR1SMN1; SMN2HSD17B10ALDH1A1
SCHEMBL30672471 0.78 MERTK (0.47) MERTKSMN1; SMN2HSD17B10ALDH1A1KDM4E
SCHEMBL30672525 0.78 TGFBR1 (0.39) SMN1; SMN2ALDH1A1KDM4EHPGDMARS1
SCHEMBL30185699 0.77 HPGD (0.49) NPSR1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL30672112 0.76 MKNK1 (0.46) MAPK1ALDH1A1KDM4EHPGDMAT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3436461-B1 PYRROLOTRIAZINE COMPOUNDS AS TAM INHIBITORS INCYTE CORP (US) 2023-11-01 EP disclosed