SCHEMBL30690765

SCHEMBL30690765

Cc1ncc(NC(=O)CN2CCC[C@@H]2C)cc1NC(=O)c1cnc2c(c1)cc(C1=CCOCC1)n2COCC[Si](C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.34
GSK3B P49841 4/20 0.32
DYRK1A Q13627 4/20 0.32
WNT1 P04628 3/20 0.32
HDAC3 O15379 2/20 0.31
HDAC1 Q13547 2/20 0.31
HDAC2 Q92769 2/20 0.31
MCHR1 Q99705 1/20 0.31
RECQL P46063 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30690687 0.87 PIK3CA (0.32) HDAC3HDAC1HDAC2
SCHEMBL30690763 0.87 GSK3B (0.36) HRH3GSK3BDYRK1AWNT1HDAC3
SCHEMBL30690797 0.86 GSK3B (0.44) HRH3GSK3BDYRK1AWNT1HDAC3
SCHEMBL30690779 0.84 GSK3B (0.35) HRH3GSK3BDYRK1AWNT1HDAC3
SCHEMBL30690782 0.84 ABL1 (0.32) HDAC3HDAC1HDAC2
SCHEMBL30690780 0.82 HDAC3 (0.34) HDAC3HDAC1HDAC2
SCHEMBL30690482 0.81 KIT (0.41) HRH3GSK3BDYRK1AWNT1RECQL
SCHEMBL30690691 0.76 AURKB (0.37) HRH3GSK3BDYRK1AWNT1
SCHEMBL30690504 0.75 HRH3 (0.39) HRH3GSK3BDYRK1AWNT1MCHR1
SCHEMBL30690792 0.75 PIK3CD (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023247593-A1 PYRROLOPYRIDINE CARBOXAMIDES AND THEIR USES AS PDGFR INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2023-12-28 WO disclosed