SCHEMBL30697102

SCHEMBL30697102

CCOC(=O)c1ncc(C)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JMJD6 Q6NYC1 1/20 0.43
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPC1 O15118 3/20 0.41
ALDH1A1 P00352 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
XBP1 P17861 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TLR9 Q9NR96 1/20 0.41
RAB9A P51151 2/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20399682 1.00 JMJD6 (0.43) JMJD6CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL24880001 0.89 ALDH1A1 (0.40) JMJD6ALDH1A1MAPTGABRA1GABRG2
SCHEMBL29664441 0.87 THRB (0.43) JMJD6CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL4018903 0.87 THRB (0.43) JMJD6CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL15968597 0.85 CA12 (0.46) JMJD6CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL6559030 0.85 TSHR (0.47) CYP2C9CYP2C19NPC1ALDH1A1NPSR1
SCHEMBL29859779 0.85 TSHR (0.47) CYP2C9CYP2C19NPC1ALDH1A1NPSR1
SCHEMBL7684716 0.84 S1PR1 (0.49) JMJD6CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL17362538 0.84 TARBP2 (0.42) JMJD6CYP2C9CYP2C19NPC1ALDH1A1
SCHEMBL15431711 0.83 ATM (0.47) NPC1ALDH1A1NPSR1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119451961-A Carboxamide derivative with RSK inhibition effect, pharmaceutical composition containing carboxamide derivative and application of carboxamide derivative 广州科恩泰生物医药科技有限公司 2025-02-14 CN disclosed
CN-117186098-A Carboxamide derivative with RSK inhibition effect, pharmaceutical composition containing carboxamide derivative and application of carboxamide derivative 上海科恩泰生物医药科技有限公司 2023-12-08 CN disclosed