SCHEMBL30714742

SCHEMBL30714742

CN1CCC(NC(=O)c2c3cc(OCc4ccnn4C)ccc3nn2C)C1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 10/20 0.40
CHRNB2 P17787 5/20 0.40
CHRNA4 P43681 5/20 0.40
GUCY1B2 O75343 1/20 0.38
GUCY1A2 P33402 1/20 0.38
GUCY1A1 Q02108 1/20 0.38
GUCY1B1 Q02153 1/20 0.38
CHRNB4 P30926 3/20 0.38
CHRNA3 P32297 3/20 0.38
HTR3A P46098 1/20 0.37
CD38 P28907 1/20 0.37
DRD4 P21917 1/20 0.37
SLC6A2 P23975 1/20 0.37
KCNH2 Q12809 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30714613 0.88 CD38 (0.40) SLC6A5CD38
SCHEMBL30714713 0.86 HTR3A (0.51) SLC6A5HTR3A
SCHEMBL30714662 0.82 CYP11B2 (0.33) HTR3A
SCHEMBL30714614 0.82 GUCY1B2 (0.40) SLC6A5CHRNB2CHRNA4GUCY1B2GUCY1A2
SCHEMBL30714756 0.82 HPGDS (0.43) RAB9A
SCHEMBL30714709 0.81 SSTR4 (0.43) SLC6A5CHRNB2CHRNA4GUCY1B2GUCY1A2
SCHEMBL30714689 0.81 HPGDS (0.35) HTR3A
SCHEMBL30714618 0.81 SCN9A (0.37) HTR3A
SCHEMBL30714550 0.80 KDM4E (0.46) SLC6A5HTR3ADRD4
SCHEMBL26696010 0.79 HPGDS (0.41) KCNH2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS UNIV LEUVEN KATH (BE) 2025-12-11 US disclosed
CN-119968362-A Indazole derivatives for the treatment of TRPM3 mediated disorders 勒芬天主教大学 2025-05-09 CN disclosed
EP-4499624-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS Katholieke Universiteit Leuven KU Leuven Research & Development (BE) 2025-02-05 EP disclosed
WO-2023230540-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS TRPV3, TRPM2, TRPV1 SLC6A5 904/4885CHRNB2 482/4885CHRNA4 393/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.