SCHEMBL30719630

SCHEMBL30719630

Cc1cc(-c2cn(C(=O)OC(C)(C)C)c3ccccc23)ccc1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.53
PIM1 P11309 1/20 0.47
MARK3 P27448 1/20 0.47
MAP4K2 Q12851 1/20 0.47
CAMK2B Q13554 1/20 0.47
PIM3 Q86V86 1/20 0.47
PIM2 Q9P1W9 1/20 0.47
BRD4 O60885 2/20 0.45
CREBBP Q92793 2/20 0.45
EPHX1 P07099 1/20 0.44
HTR6 P50406 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
PDE10A Q9Y233 1/20 0.42
ACHE P22303 1/20 0.41
HTT P42858 1/20 0.40
NR1H2 P55055 2/20 0.37
TLR8 Q9NR97 1/20 0.36
BRPF1 P55201 1/20 0.36
BRD9 Q9H8M2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23496956 1.00 L3MBTL1 (0.53) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL27257521 0.82 L3MBTL1 (0.53) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL5871186 0.81 L3MBTL1 (0.51) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL30620463 0.80 L3MBTL1 (0.50) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL31070592 0.79 L3MBTL1 (0.47) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL21246906 0.78 L3MBTL1 (0.59) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL1196432 0.78 L3MBTL1 (0.62) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL22468928 0.78 KMT2A (0.49) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL29831138 0.76 L3MBTL1 (0.47) L3MBTL1PIM1MARK3MAP4K2CAMK2B
SCHEMBL23330849 0.76 L3MBTL1 (0.47) L3MBTL1PIM1MARK3MAP4K2CAMK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117586108-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN claimed
CN-117586191-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN disclosed
CN-117586108-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-02-23 CN disclosed
CN-111542515-B TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2023-12-05 CN disclosed