SCHEMBL30720875

SCHEMBL30720875

C[Si](C)(C)CCOCn1cnc(Cl)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
DGAT1 O75907 5/20 0.37
POLB P06746 1/20 0.36
PKM P14618 1/20 0.35
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13560502 0.81 DGAT1 (0.35) MAPTNPSR1DGAT1
SCHEMBL3635281 0.80 DGAT1 (0.35) MAPTNPSR1DGAT1BRD4CREBBP
SCHEMBL3028008 0.79 DGAT1 (0.38) MAPTDGAT1POLBPKM
SCHEMBL28841318 0.78 DGAT1 (0.37) MAPTNPSR1DGAT1BRD4CREBBP
SCHEMBL31340868 0.76 FDPS (0.45)
SCHEMBL357273 0.76 FDPS (0.45)
SCHEMBL31138390 0.76 DGAT1 (0.36) MAPTDGAT1
SCHEMBL9928488 0.76 DGAT1 (0.36) MAPTDGAT1
SCHEMBL3267555 0.76 P2RX7 (0.43) MAPTDGAT1
SCHEMBL12620882 0.76 ADORA2A (0.37) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4739393-A1 TETRAHYDROQUINAZOLINE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS Merck Sharp & Dohme LLC (US) 2026-05-13 EP disclosed
EP-4642782-A2 ALPHA-V-BETA-8 INTEGRIN INHIBITORS AND USES THEREOF Pliant Therapeutics, Inc. (US) 2025-11-05 EP disclosed
EP-4554933-A1 HERBICIDAL IMIDAZOLE COMPOUNDS Syngenta Crop Protection AG (CH) 2025-05-21 EP disclosed
WO-2025072539-A1 AMINO ACID COMPOUNDS WITH NITROGEN LINKERS AND USES THEREOF PLIANT THERAPEUTICS, INC. (US) 2025-04-03 WO disclosed
CN-119451949-A Herbicidal imidazole compounds 先正达农作物保护股份公司 2025-02-14 CN disclosed
US-20250026759-A1 TETRAHYDROQUINAZOLINE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS MERCK SHARP & DOHME LLC (US) 2025-01-23 US disclosed
WO-2025014788-A1 TETRAHYDROQUINAZOLINE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS MERCK SHARP & DOHME LLC (US) 2025-01-16 WO disclosed
WO-2024013018-A1 HERBICIDAL IMIDAZOLE COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2024-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250026759-A1 TETRAHYDROQUINAZOLINE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS ACIN1, REV1, NFATC1 MAPT 2556/4885NPSR1 4707/4885DGAT1 3822/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.