SCHEMBL30724683

SCHEMBL30724683

Cc1ccnc(NC2Cc3ccc(Br)cc3C2)n1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 11/20 0.41
GBA1 P04062 1/20 0.41
CYP2C8 P10632 2/20 0.39
CYP2C9 P11712 2/20 0.39
KCNH2 Q12809 2/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2D6 P10635 1/20 0.39
HDAC6 Q9UBN7 3/20 0.38
ADRA2A P08913 1/20 0.36
PNMT P11086 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30724692 0.87 HDAC8 (0.41) HDAC8HDAC6
SCHEMBL30724695 0.83 HDAC8 (0.50) HDAC8GBA1HDAC6ADRA2APNMT
SCHEMBL30798351 0.82 HDAC8 (0.42) HDAC8CYP2C9KCNH2CYP2D6
SCHEMBL28658090 0.74 GBA1 (0.39) HDAC8GBA1CYP2C8CYP2C9KCNH2
SCHEMBL91469 0.74 CTSK (0.49) CYP2C9
SCHEMBL91478 0.71 CTSK (0.58)
SCHEMBL30724677 0.71 GBA1 (0.42) HDAC8GBA1HDAC6ADRA2APNMT
SCHEMBL30724682 0.70 HDAC8 (0.54) HDAC8GBA1HDAC6
SCHEMBL91484 0.70 CTSK (0.60)
SCHEMBL12367075 0.70 IKBKB (0.61) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396471-A Novel piperidine derivatives and pharmaceutical compositions for inhibiting autotaxin comprising the same 株式会社次代生物科学 2024-01-12 CN disclosed