SCHEMBL30724677

SCHEMBL30724677

Clc1ccnc(NC2Cc3ccc(Br)cc3C2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.42
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
PRMT5 O14744 1/20 0.39
HRH4 Q9H3N8 2/20 0.37
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
ADRA2A P08913 1/20 0.34
PNMT P11086 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
PHGDH O43175 1/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30724682 0.80 HDAC8 (0.54) GBA1NOS2HRH4HDAC8HDAC6
SCHEMBL30724688 0.79 GBA1 (0.47) GBA1PRMT5HDAC8HDAC6ADRA2A
SCHEMBL30724695 0.75 HDAC8 (0.50) GBA1HDAC8HDAC6KDM4EADRA2A
SCHEMBL27195343 0.74 SORT1 (0.42) GBA1PRMT5HDAC8HDAC6
SCHEMBL30724674 0.74 SORT1 (0.42) GBA1PRMT5HDAC8HDAC6
SCHEMBL24112178 0.71 MAPK1 (0.39) GBA1PRMT5HDAC8HDAC6MCHR1
SCHEMBL24112177 0.71 MAPK1 (0.39) GBA1PRMT5HDAC8HDAC6MCHR1
SCHEMBL30724683 0.71 HDAC8 (0.41) GBA1HDAC8HDAC6ADRA2APNMT
SCHEMBL24613289 0.70 PNMT (0.44) GBA1PRMT5ADRA2APNMTADRA2B
SCHEMBL3576035 0.70 NOS1 (0.52) NOS1NOS2HRH4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396471-A Novel piperidine derivatives and pharmaceutical compositions for inhibiting autotaxin comprising the same 株式会社次代生物科学 2024-01-12 CN disclosed