SCHEMBL30728873

SCHEMBL30728873

COc1cccc(-c2cccc(CBr)c2OC)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.43
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2D6 P10635 3/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2C19 P33261 3/20 0.42
CYP1A1 P04798 2/20 0.42
CYP2E1 P05181 2/20 0.42
CYP2C8 P10632 2/20 0.42
CYP2A6 P11509 2/20 0.42
CYP4B1 P13584 2/20 0.42
CYP2B6 P20813 2/20 0.42
CYP3A5 P20815 2/20 0.42
CYP2A7 P20853 2/20 0.42
CYP3A7 P24462 2/20 0.42
CYP2F1 P24903 2/20 0.42
CYP2C18 P33260 2/20 0.42
CYP2J2 P51589 2/20 0.42
CYP4F2 P78329 2/20 0.42
CYP4F8 P98187 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28854331 0.87 HTR7 (0.51) HTR7CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28517574 0.84 ABL1 (0.46) HTR7CLK4ABCB1
SCHEMBL20957481 0.83 PDCD1 (0.44) HTR7CYP2A6ALDH1A1CD274MAPK1
SCHEMBL2020140 0.75 ABL1 (0.59) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9078093 0.75 ALDH1A1 (0.40) ALDH1A1ABCB1TSHRMAPK1
SCHEMBL8279410 0.74 MGAT2 (0.57) HTR7CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3388700 0.74 MAPK1 (0.46) HTR7CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL12490805 0.73 MGAT2 (0.56) HTR7CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL14318443 0.73 SMARCA2 (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5094201 0.73 FNTA (0.53) CYP1A2CYP3A4CYP2D6CYP2C19CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117186001-B AHA1 inhibitor with multiple myeloma-resisting activity and preparation method and application thereof 南京中医药大学 2024-09-17 CN disclosed
CN-117186001-A AHA1 inhibitor with multiple myeloma-resisting activity and preparation method and application thereof 南京中医药大学 2023-12-08 CN disclosed