SCHEMBL30729987

SCHEMBL30729987

CCSc1ncc2[nH]cnc2n1.[Sn]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
POLA1 P09884 1/20 0.40
CDK2 P24941 4/20 0.39
RXFP1 Q9HBX9 1/20 0.39
PAK1 Q13153 2/20 0.37
F7 P08709 1/20 0.35
F3 P13726 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
CDK1 P06493 3/20 0.33
CCNB1 P14635 3/20 0.33
CCNT1 O60563 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
CCNH P51946 1/20 0.33
HASPIN Q8TF76 1/20 0.33
QPCT Q16769 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7592034 0.98 ALDH1A1 (0.49) ALDH1A1KDM4EPOLA1CDK2RXFP1
SCHEMBL27535767 0.83 XDH (0.47) ALDH1A1KDM4EPOLA1CDK2RXFP1
SCHEMBL10923939 0.80 XDH (0.49) ALDH1A1KDM4EPOLA1PAK1CYP1A2
SCHEMBL1371022 0.79 ALDH1A1 (0.53) ALDH1A1KDM4EPOLA1CDK2RXFP1
SCHEMBL11802315 0.78 ALDH1A1 (0.57) ALDH1A1KDM4EPOLA1CDK2RXFP1
SCHEMBL2563787 0.78 ALDH1A1 (0.45) ALDH1A1KDM4EPOLA1CDK2RXFP1
SCHEMBL6833311 0.76 F7 (0.43) ALDH1A1F7F3CYP1A2HASPIN
SCHEMBL11500976 0.76 ALDH1A1 (0.47) ALDH1A1KDM4EPOLA1CDK2RXFP1
SCHEMBL29120496 0.75 KDM4E (0.58) ALDH1A1KDM4EPOLA1CDK2RXFP1
SCHEMBL28715732 0.75 ALDH1A1 (0.58) ALDH1A1KDM4EPOLA1CDK2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117769554-A Small molecule inhibitors of KRAS muteins 大鹏药品工业株式会社 2024-03-26 CN disclosed
CN-117396472-A SOS1 inhibitors and uses thereof 上海齐鲁锐格医药研发有限公司 2024-01-12 CN disclosed