SCHEMBL30730775

SCHEMBL30730775

CCOC(=O)c1cc2c(-c3cncc(-c4ccc(N5CCCC5=O)cc4)c3)ccnc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.41
HSD17B10 Q99714 1/20 0.41
BRAF P15056 1/20 0.41
NUDT1 P36639 2/20 0.41
DGAT2 Q96PD7 1/20 0.40
TBK1 Q9UHD2 1/20 0.40
MMP13 P45452 3/20 0.40
NPC1 O15118 1/20 0.40
MMP2 P08253 2/20 0.39
MMP14 P50281 2/20 0.39
LMNA P02545 1/20 0.37
TNIK Q9UKE5 1/20 0.36
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP11B2 P19099 1/20 0.35
CD38 P28907 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22553840 1.00 PKM (0.41) PKMHSD17B10BRAFNUDT1DGAT2
SCHEMBL30731117 0.92 NUDT1 (0.43) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL22553938 0.92 NUDT1 (0.43) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL30730826 0.92 NUDT1 (0.43) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL30730786 0.89 NUDT1 (0.41) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL22553907 0.89 NUDT1 (0.41) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL22553975 0.87 TBK1 (0.44) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL30730801 0.87 TBK1 (0.44) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL22554135 0.86 NUDT1 (0.57) PKMNUDT1DGAT2TBK1NPC1
SCHEMBL30731110 0.86 NUDT1 (0.46) NUDT1DGAT2TBK1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN claimed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed