SCHEMBL30737241

SCHEMBL30737241

COC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCOCCOCCOCCOCCN)cccc23)nc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.37
HDAC1 Q13547 3/20 0.37
POLB P06746 1/20 0.36
KMT2A Q03164 2/20 0.35
PRKCD Q05655 2/20 0.35
CAMK2B Q13554 2/20 0.35
CAMK2G Q13555 2/20 0.35
AURKB Q96GD4 2/20 0.35
MEN1 O00255 1/20 0.35
HIF1A Q16665 1/20 0.35
TSHR P16473 1/20 0.35
HPGD P15428 2/20 0.35
DAPK3 O43293 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
CHEK2 O96017 1/20 0.35
PHKG2 P15735 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CLK2 P49760 1/20 0.35
IRAK1 P51617 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30737086 0.88 PLK1 (0.38) POLBKMT2A
SCHEMBL30737162 0.87 F2 (0.41) HDAC3HDAC1POLBKMT2AMEN1
SCHEMBL30737153 0.82 HCAR3 (0.38) POLBKMT2AMEN1ALDH1A1KDM4E
SCHEMBL30737309 0.80 GABRA5 (0.41) HPGDKDM4EMAPT
SCHEMBL30737273 0.76 PLK1 (0.47) KMT2AAURKBMEN1PIM2AURKA
SCHEMBL30737232 0.74 HCAR3 (0.41) KMT2AMEN1ALDH1A1KDM4EMAPT
SCHEMBL31646525 0.72 LOXL2 (0.55) KMT2AMEN1ALDH1A1MAPTSMN1; SMN2
SCHEMBL30737488 0.69 MAPT (0.45) KMT2AMEN1TSHRHPGDALDH1A1
SCHEMBL30737383 0.69 MAPT (0.45) KMT2AMEN1TSHRHPGDALDH1A1
SCHEMBL30737283 0.67 PLK1 (0.45) AURKBAURKALCKKDRTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4543858-A1 BIFUNCTIONAL MOLECULES THAT SELECTIVELY INDUCE DEGRADATION OF EXTRACELLULAR TARGETS IN LYSOSOMES Draupnir Bio ApS (DK) 2025-04-30 EP disclosed
WO-2023247754-A1 BIFUNCTIONAL MOLECULES THAT SELECTIVELY INDUCE DEGRADATION OF EXTRACELLULAR TARGETS IN LYSOSOMES DRAUPNIR BIO APS (DK) 2023-12-28 WO disclosed