SCHEMBL30744362

SCHEMBL30744362

NCc1cn(Cc2ccc(C(F)(F)F)nc2)cn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.37
GRIN1 Q05586 2/20 0.36
GRIN2B Q13224 2/20 0.36
LOXL2 Q9Y4K0 2/20 0.36
DAO P14920 3/20 0.35
PPARD Q03181 1/20 0.35
LOX P28300 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
CPB1 P15086 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
KCNH2 Q12809 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
PRMT5 O14744 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21491764 1.00 TRPV4 (0.37) TRPV4GRIN1GRIN2BLOXL2DAO
SCHEMBL28517068 0.80 PPARD (0.39) PPARDMAOBCPB1JAK2JAK1
SCHEMBL21492711 0.80 PPARD (0.42) PPARDKDM1AMAOAMAOBKCNH2
SCHEMBL21492945 0.77 CYP11B1 (0.36) TRPV4GRIN1GRIN2BDAOPPARD
SCHEMBL28524266 0.77 CYP2C19 (0.38) TRPV4GRIN1GRIN2BDAOPPARD
SCHEMBL24208607 0.77 CPB1 (0.39) TRPV4GRIN1GRIN2BDAOPPARD
SCHEMBL30744491 0.77 CYP11B1 (0.36) TRPV4GRIN1GRIN2BDAOPPARD
SCHEMBL21503682 0.76 LOXL2 (0.40) TRPV4GRIN1GRIN2BLOXL2DAO
Hydrochloric Acid SCHEMBL21491894 0.75 LMNA (0.41) TRPV4GRIN1GRIN2BLOXL2DAO
Hydrochloric Acid SCHEMBL30744436 0.75 LMNA (0.41) TRPV4GRIN1GRIN2BLOXL2DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-B Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2024-03-12 CN disclosed