SCHEMBL30786118

SCHEMBL30786118

C(=C/c1nn(C2CCCCO2)c2ccccc12)\c1ccc(CN2CCCC2)cn1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 3/20 0.34
PRKCD Q05655 3/20 0.34
ACHE P22303 2/20 0.33
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
PDE1B Q01064 2/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
CNR2 P34972 1/20 0.32
DRD4 P21917 1/20 0.32
CDK4 P11802 1/20 0.31
CDK6 Q00534 1/20 0.31
HRH3 Q9Y5N1 2/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30786116 0.88 RXRA (0.33) PRKCQPRKCDACHERXRARXRB
SCHEMBL30786199 0.88 CYP4F2 (0.35) PRKCQPRKCDRXRARXRBRXRG
SCHEMBL30786077 0.84 RXRA (0.32) RXRARXRBRXRG
SCHEMBL30786167 0.82 PSEN1 (0.36) RXRARXRBRXRGHRH3
SCHEMBL31475223 0.82 FAAH (0.34) PRKCQPRKCDRXRARXRBRXRG
SCHEMBL30786228 0.81 PDCD1 (0.37) PRKCQPRKCDACHEPDCD1CD274
SCHEMBL31517065 0.80 FAAH (0.37) PRKCQPRKCDKDR
SCHEMBL30786196 0.80 KDR (0.43) KDR
SCHEMBL31517057 0.80 KDM4E (0.34) PDE1B
SCHEMBL29705188 0.80 FGFR1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024032584-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF 苏州必扬医药科技有限公司 2024-02-15 WO disclosed