SCHEMBL30786127

SCHEMBL30786127

Cc1ncc(CN2CCCC2)cc1/C=C/c1nn(C2CCCCO2)c2cc(Oc3ccccc3C(=O)O)ccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
DRD1 P21728 1/20 0.35
KCNH2 Q12809 1/20 0.32
MCHR1 Q99705 1/20 0.32
CCR8 P51685 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALOX5AP P20292 2/20 0.31
PPARG P37231 1/20 0.31
DGAT1 O75907 1/20 0.31
HRH2 P25021 2/20 0.31
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
AGTR1 P30556 1/20 0.31
AGTR2 P50052 1/20 0.31
CCR3 P51677 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30786167 0.90 PSEN1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL31517057 0.84 KDM4E (0.34) KCNH2MCHR1CCR8KDM4ECCR3
SCHEMBL31475223 0.75 FAAH (0.34) MCHR1MEN1KMT2A
SCHEMBL31517065 0.72 FAAH (0.37) MCHR1KDM4EMEN1ALDH1A1KMT2A
SCHEMBL30786118 0.71 PRKCQ (0.34)
SCHEMBL30786196 0.71 KDR (0.43) KMT2A
SCHEMBL30786199 0.70 CYP4F2 (0.35) CYP4F2CYP4A11
SCHEMBL30786116 0.70 RXRA (0.33) ALDH1A1
SCHEMBL177618 0.69 KDM4E (0.43) KDM4EALOX5APCYP4F2CYP4A11ALDH1A1
SCHEMBL2237687 0.69 KDM4E (0.43) KDM4EALOX5APCYP4F2CYP4A11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024032584-A1 PROTEIN TYROSINE KINASE INHIBITOR AND MEDICAL USE THEREOF 苏州必扬医药科技有限公司 2024-02-15 WO disclosed