SCHEMBL30801775

SCHEMBL30801775

O=C1[C@H]2CNCCN2CCN1c1cccc(-c2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.49
HTR7 P34969 3/20 0.49
ALDH1A1 P00352 4/20 0.40
USP2 O75604 3/20 0.40
TP53 P04637 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 3/20 0.40
HSD17B10 Q99714 3/20 0.40
MAPK1 P28482 2/20 0.40
CYP3A4 P08684 2/20 0.40
TSHR P16473 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
HSD11B1 P28845 2/20 0.39
HIF1A Q16665 1/20 0.39
MGLL Q99685 2/20 0.38
FAAH O00519 1/20 0.38
HSP90AA1 P07900 1/20 0.38
PKM P14618 1/20 0.38
HTT P42858 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30801844 0.85 DRD2 (0.49) HTR1AHTR7ALDH1A1TP53CYP1A2
SCHEMBL30801761 0.81 COMT (0.38) HTR1AHTR7TAAR1HTR2AHTR2C
SCHEMBL30801864 0.81 ALDH1A1 (0.51) HTR7ALDH1A1TSHRHTR2AHTR2C
SCHEMBL30801822 0.78 LTA4H (0.49) ALDH1A1TAAR1MGLLHTR2AHTR2C
SCHEMBL30801833 0.77 F10 (0.40) TAAR1MGLLHTR2AHTR2CHTR2B
SCHEMBL30801829 0.77 SLC6A2 (0.51) HTR1AALDH1A1CYP1A2CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL3609828 0.76 SLC6A2 (0.39) HTR1AHTR7TAAR1HTR6HTR2A
Hydrochloric Acid SCHEMBL3609734 0.76 TAAR1 (0.42) ALDH1A1TAAR1HTR2AHTR2CHTR2B
SCHEMBL23574003 0.76 USP30 (0.46) ALDH1A1MGLLFAAHHSP90AA1PKM
SCHEMBL30801882 0.76 USP30 (0.46) ALDH1A1MGLLFAAHHSP90AA1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3793997-B1 FUSED BICYCLIC COMPOUNDS USEFUL AS UBIQUITIN-SPECIFIC PEPTIDASE 30 INHIBITORS FORMA THERAPEUTICS INC (US) 2024-03-13 EP claimed