SCHEMBL30820765

SCHEMBL30820765

Fc1cnccc1-c1cncc2c1OCC2

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.37
PDE4B Q07343 2/20 0.36
CDC7 O00311 1/20 0.35
RIPK1 Q13546 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
RPS6KA3 P51812 2/20 0.32
MELK Q14680 1/20 0.32
RPS6KA2 Q15349 1/20 0.32
RPS6KA1 Q15418 1/20 0.32
CYP1A2 P05177 1/20 0.32
METAP2 P50579 1/20 0.32
PARP1 P09874 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
BUB1 O43683 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29677390 0.78 PDE4B (0.34) PDE4BSIGMAR1RPS6KA3CYP1A2PARP1
SCHEMBL30820792 0.77 PDE4B (0.36) PDE4BPARP1
SCHEMBL31301232 0.72 NUDT1 (0.57) NUDT1CDC7RPS6KA3CYP1A2METAP2
SCHEMBL30820691 0.68 PDE4B (0.32) PDE4BRPS6KA3CYP1A2
SCHEMBL4067954 0.67 SIGMAR1 (0.39) SIGMAR1RPS6KA3
SCHEMBL15466341 0.67 MAOA (0.41) SIGMAR1CYP1A2
SCHEMBL30820819 0.67 DYRK1A (0.40) PDE4BCDC7MKNK1MKNK2
SCHEMBL30820814 0.67 DYRK1A (0.40) CDC7
SCHEMBL31033492 0.65
SCHEMBL125109 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12534474-B2 Dihydrofuropyridine derivatives as rho-kinase inhibitors CHIESI FARMACEUTICI S.P.A. (IT) 2026-01-27 US disclosed
US-20240092792-A1 DIHYDROFUROPYRIDINE DERIVATIVES AS RHO- KINASE INHIBITORS CHIESI FARMACEUTICI S.P.A. (IT) 2024-03-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240092792-A1 DIHYDROFUROPYRIDINE DERIVATIVES AS RHO- KINASE INHIBITORS ROCK1, ROCK2, RHOA NUDT1 261/4885PDE4B 22/4885CDC7 738/4885
US-12534474-B2 Dihydrofuropyridine derivatives as rho-kinase inhibitors ROCK1, RHOC, ROCK2 NUDT1 288/4885PDE4B 54/4885CDC7 509/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.