SCHEMBL30833278

SCHEMBL30833278

CN1C(=O)CC(=O)c2cc(I)ccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.57
TDP2 O95551 2/20 0.37
OPRK1 P41145 2/20 0.36
PDE4D Q08499 1/20 0.36
GAA P10253 2/20 0.35
LMNA P02545 1/20 0.35
TSPO P30536 1/20 0.35
TRIM24 O15164 1/20 0.35
APP P05067 1/20 0.34
GABRA1 P14867 3/20 0.34
GABRG2 P18507 3/20 0.34
GABRB3 P28472 3/20 0.34
GABRA5 P31644 3/20 0.34
GABRA3 P34903 3/20 0.34
GABRA2 P47869 3/20 0.34
GABRB2 P47870 3/20 0.34
GABRP O00591 2/20 0.34
GABRD O14764 2/20 0.34
GABRB1 P18505 2/20 0.34
GABRA4 P48169 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30099722 0.79 GABRA1 (0.48) OPRK1PDE4DGAALMNATSPO
SCHEMBL16506973 0.79 TRIM24 (0.49) CASP3GAALMNATRIM24ALDH1A1
SCHEMBL2759567 0.76 CASP3 (0.53) CASP3TDP2GAALMNATSPO
SCHEMBL19657308 0.75 CASP3 (0.43) CASP3TDP2OPRK1PDE4DGAA
SCHEMBL8054672 0.74 TTR (0.52) CASP3OPRK1PDE4DLMNAGABRA1
SCHEMBL5118034 0.73 CASP3 (1.00) CASP3APPALDH1A1
SCHEMBL13539267 0.72 CASP3 (0.49) CASP3TDP2GAAGABRA1GABRG2
SCHEMBL8554279 0.70 CYP11B2 (0.51) CASP3TRIM24
SCHEMBL9158816 0.70 CASP3 (0.46) CASP3GAAGABRA1GABRG2GABRB3
SCHEMBL24677008 0.69 PDE3B (0.44) LMNAGABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117580829-A Quinoline and azaquinolines as inhibitors of CD38 勃林格英格翰国际有限公司 2024-02-20 CN disclosed