SCHEMBL30833672

SCHEMBL30833672

NS(=O)(=O)Cc1ccccc1Nc1nc(Nc2ccc3c(N4CCOCC4)n[nH]c3c2)ncc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 5/20 0.51
MAPK9 P45984 4/20 0.50
MAPK10 P53779 4/20 0.50
MAPK8 P45983 2/20 0.50
EGFR P00533 2/20 0.49
CCNK O75909 1/20 0.49
CCNA2 P20248 1/20 0.49
CDK2 P24941 1/20 0.49
CCND3 P30281 1/20 0.49
CDK9 P50750 1/20 0.49
CDK6 Q00534 1/20 0.49
PKMYT1 Q99640 2/20 0.49
AXL P30530 1/20 0.49
INSR P06213 1/20 0.49
IGF1R P08069 1/20 0.49
PTK2 Q05397 1/20 0.49
PTK2B Q14289 1/20 0.49
SLC2A1 P11166 1/20 0.48
ULK1 O75385 1/20 0.47
MAP3K7 O43318 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833699 0.87 EGFR (0.49) ALKMAPK9MAPK10MAPK8EGFR
SCHEMBL29190617 0.86 ALK (0.68) ALKMAPK9MAPK10EGFRCCNK
SCHEMBL30833696 0.85 ALK (0.52) ALKMAPK9MAPK10PTK2ULK1
SCHEMBL30833666 0.83 ALK (0.49) ALKEGFRIGF1R
SCHEMBL30833773 0.81 BRD4 (0.47) ALKEGFRCDK2PTK2PTK2B
SCHEMBL30833757 0.79 ALK (0.47) ALKCCNKCCNA2CDK2CCND3
SCHEMBL30833776 0.77 ALK (0.48) ALKPTK2
SCHEMBL30833718 0.77 JAK3 (0.47) ALKMAPK9MAPK8EGFRCDK2
SCHEMBL29190605 0.77 ALK (0.67) ALKEGFRCCNKCCNA2CDK2
SCHEMBL30833724 0.77 ALK (0.52) ALKMAPK9MAPK10MAPK8EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed