SCHEMBL30833718

SCHEMBL30833718

Cc1cnc(Nc2ccc3c(Cl)n[nH]c3c2)nc1Nc1ccccc1CS(N)(=O)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 6/20 0.47
JAK1 P23458 6/20 0.47
ALK Q9UM73 9/20 0.46
PKMYT1 Q99640 1/20 0.45
SYK P43405 2/20 0.42
IGF1R P08069 2/20 0.41
AURKA O14965 2/20 0.41
PTK2 Q05397 2/20 0.41
CDC7 O00311 1/20 0.41
PLK4 O00444 1/20 0.41
CHEK1 O14757 1/20 0.41
DCLK1 O15075 1/20 0.41
PDPK1 O15530 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
ROCK2 O75116 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
CHEK2 O96017 1/20 0.41
ABL1 P00519 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833696 0.91 ALK (0.52) ALKPTK2METFLT3MAPK9
SCHEMBL30833797 0.85 ALK (0.44) JAK3JAK1ALKPKMYT1IGF1R
SCHEMBL29190642 0.84 ALK (0.59) JAK3JAK1ALKPKMYT1EGFR
SCHEMBL30833757 0.81 ALK (0.47) ALKPTK2METCDK2FLT3
SCHEMBL30833666 0.81 ALK (0.49) ALKIGF1REGFRMETFLT3
SCHEMBL30833776 0.80 ALK (0.48) ALKSYKPTK2METFLT3
SCHEMBL30833764 0.78 IGF1R (0.45) JAK3JAK1ALKSYKIGF1R
SCHEMBL30833774 0.76 IGF1R (0.43) JAK3ALKSYKIGF1RAURKA
SCHEMBL29190551 0.76 ALK (0.67) ALKPTK2EGFRMETFLT3
SCHEMBL30833765 0.75 PKMYT1 (0.38) ALKPKMYT1IGF1RAURKAINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed