SCHEMBL30833752

SCHEMBL30833752

CN1CCN(C2CCN(c3n[nH]c4cc([N+](=O)[O-])ccc34)CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
KCNH2 Q12809 1/20 0.41
HRH4 Q9H3N8 3/20 0.40
SIRT6 Q8N6T7 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39
RHOA P61586 1/20 0.38
MAPK1 P28482 1/20 0.38
ALDH1A1 P00352 2/20 0.38
ACHE P22303 2/20 0.37
APP P05067 1/20 0.37
BCHE P06276 1/20 0.37
AURKA O14965 1/20 0.37
LMNA P02545 1/20 0.37
ALK Q9UM73 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190644 1.00 MEN1 (0.41) MEN1KMT2AKCNH2HRH4SIRT6
SCHEMBL30833799 0.89 SIRT6 (0.50) MEN1KMT2AHRH4SIRT6HRH3
SCHEMBL4784574 0.89 SIRT6 (0.50) MEN1KMT2AHRH4SIRT6HRH3
SCHEMBL29190586 0.87 MAPK1 (0.43) MEN1KMT2AHRH3RHOAMAPK1
SCHEMBL30833680 0.87 MAPK1 (0.43) MEN1KMT2AHRH3RHOAMAPK1
SCHEMBL30833677 0.87 MAPK1 (0.43) MEN1KMT2AHRH3RHOAMAPK1
SCHEMBL29190522 0.81 KCNH2 (0.44) KCNH2MAPK1
SCHEMBL30833743 0.81 KCNH2 (0.44) KCNH2MAPK1
SCHEMBL29190649 0.80 HRH4 (0.44) MEN1KMT2AKCNH2HRH4SIRT6
SCHEMBL30833658 0.80 HRH4 (0.44) MEN1KMT2AKCNH2HRH4SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed