SCHEMBL30833772

SCHEMBL30833772

Nc1cccc(Nc2ncc(Cl)c(Nc3ccccc3CN[SH](=O)=O)n2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.46
CCNA2 P20248 5/20 0.46
CDK9 P50750 4/20 0.46
CCNK O75909 3/20 0.46
CCND3 P30281 3/20 0.46
CDK6 Q00534 3/20 0.46
MAPK9 P45984 4/20 0.41
MAPK10 P53779 4/20 0.41
ALK Q9UM73 3/20 0.40
MET P08581 2/20 0.40
ULK1 O75385 1/20 0.39
IGF1R P08069 1/20 0.39
MAPK8 P45983 1/20 0.39
AURKA O14965 1/20 0.39
LRRK2 Q5S007 1/20 0.38
CTSC P53634 1/20 0.38
CDC7 O00311 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
ROCK2 O75116 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833649 0.83 CDK9 (0.47) CDK2CCNA2CDK9CCNKCCND3
SCHEMBL30833627 0.79 BCL6 (0.39) CDK2CCNA2CDK9CCNKCCND3
SCHEMBL29190618 0.78 ALK (0.59) CDK2CCNA2CDK9CCNKCCND3
SCHEMBL30833687 0.76 ALK (0.50) MAPK9MAPK10ALKMETULK1
SCHEMBL29190576 0.76 CDK2 (0.53) CDK2CCNA2CDK9CCNKCCND3
SCHEMBL30833804 0.76 CDK2 (0.53) CDK2CCNA2CDK9CCNKCCND3
SCHEMBL30833700 0.74 KDR (0.52) CDK2CDK9MAPK9MAPK10ALK
SCHEMBL30833737 0.74 CDK2 (0.42) CDK2CCNA2CDK9CCNKCCND3
SCHEMBL30833783 0.74 SYK (0.47) CDK2CCNA2CDK9CCNKCCND3
SCHEMBL30833711 0.74 CDK2 (0.42) CDK2CCNA2CDK9CCNKCCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed