SCHEMBL30833649

SCHEMBL30833649

Nc1cccc(Nc2ncc(Cl)c(Nc3ccccc3CS(N)(=O)=O)n2)n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 3/20 0.47
CCNA2 P20248 2/20 0.47
CDK2 P24941 2/20 0.47
CCNK O75909 1/20 0.47
CCND3 P30281 1/20 0.47
CDK6 Q00534 1/20 0.47
ALK Q9UM73 8/20 0.45
MET P08581 5/20 0.42
MAPK9 P45984 2/20 0.41
MAPK10 P53779 2/20 0.41
AURKA O14965 2/20 0.40
AURKB Q96GD4 1/20 0.40
CDK7 P50613 2/20 0.40
ULK1 O75385 1/20 0.40
INSR P06213 1/20 0.40
MAPK8 P45983 1/20 0.40
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833772 0.83 CDK2 (0.46) CDK9CCNA2CDK2CCNKCCND3
SCHEMBL29190618 0.81 ALK (0.59) CDK9CCNA2CDK2CCNKCCND3
SCHEMBL30833643 0.80 ALK (0.43) CDK9ALKMETMAPK9MAPK10
SCHEMBL29190576 0.77 CDK2 (0.53) CDK9CCNA2CDK2CCNKCCND3
SCHEMBL30833804 0.77 CDK2 (0.53) CDK9CCNA2CDK2CCNKCCND3
SCHEMBL14889458 0.76 ALK (0.50) ALKMETMAPK9MAPK10
SCHEMBL30833724 0.75 ALK (0.52) CDK9CDK2ALKMETMAPK9
SCHEMBL26906809 0.71 ALK (0.48) CDK9CCNA2CDK2CCNKCCND3
SCHEMBL29904714 0.71 ALK (0.48) CDK9CCNA2CDK2CCNKCCND3
SCHEMBL30833733 0.69 PIN1 (0.36) CDK9ALKAURKAAURKBCDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed