SCHEMBL30855029

SCHEMBL30855029

COCCOc1cccc(CNc2ncco2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.47
RPS6KB1 P23443 1/20 0.47
ROCK2 O75116 4/20 0.42
ROCK1 Q13464 3/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
GAA P10253 1/20 0.40
CYP2D6 P10635 3/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
MAPK1 P28482 1/20 0.39
F2 P00734 1/20 0.39
EGFR P00533 2/20 0.39
IGF1R P08069 2/20 0.39
AURKB Q96GD4 1/20 0.38
ADORA3 P0DMS8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30855014 0.87 MTNR1A (0.53) KDM4EALDH1A1MTNR1AMTNR1BGAA
SCHEMBL25046109 0.76 BCHE (0.58) AURKARPS6KB1KDM4EALDH1A1GAA
SCHEMBL24163604 0.76 FFAR1 (0.43) ROCK1KDM4EALDH1A1CYP1A2MEN1
SCHEMBL22191536 0.75 AURKA (0.49) AURKARPS6KB1ROCK2ROCK1KDM4E
SCHEMBL17790188 0.75 KDM4E (0.51) AURKARPS6KB1ROCK2ROCK1KDM4E
SCHEMBL30854997 0.75 PPARA (0.41) ROCK2ROCK1KDM4EALDH1A1
SCHEMBL30854977 0.75 ROCK2 (0.49) AURKARPS6KB1ROCK2ROCK1KDM4E
SCHEMBL7046408 0.73 FABP1 (0.50) KDM4EALDH1A1CYP2D6CYP3A4CYP1A2
SCHEMBL28971693 0.73 CLK4 (0.52) KDM4EGAAEGFRIGF1RMEN1
SCHEMBL25302034 0.73 CHRM2 (0.59) KDM4EALDH1A1MAPK1MEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117916237-A Amino aryl integrin agonist compounds 德克萨斯心脏研究所 2024-04-19 CN claimed
CN-117916237-A Amino aryl integrin agonist compounds 德克萨斯心脏研究所 2024-04-19 CN disclosed