SCHEMBL30855014

SCHEMBL30855014

COc1cccc(CNc2ncco2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.53
MTNR1B P49286 1/20 0.53
EGFR P00533 2/20 0.48
IGF1R P08069 2/20 0.48
MAPT P10636 4/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
ALDH1A1 P00352 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
TSHR P16473 2/20 0.48
CYP2C19 P33261 2/20 0.48
TP53 P04637 2/20 0.48
HTT P42858 2/20 0.48
MAPK1 P28482 2/20 0.48
USP2 O75604 1/20 0.48
CYP2C9 P11712 1/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30855029 0.87 AURKA (0.47) MTNR1AMTNR1BEGFRIGF1RMAPT
SCHEMBL28971693 0.82 CLK4 (0.52) EGFRIGF1RMAPTMEN1KMT2A
SCHEMBL24163604 0.80 FFAR1 (0.43) MAPTMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL7046408 0.77 FABP1 (0.50) EGFRIGF1RMAPTMEN1KMT2A
SCHEMBL30855353 0.77 MTNR1A (0.55) MTNR1AMTNR1BMAPTSMN1; SMN2ALDH1A1
SCHEMBL29890148 0.77 APLNR (0.55) MEN1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL24097802 0.77 APLNR (0.55) MEN1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL20773126 0.75 HTR1B (0.49) CHRM2CHRM1CHRM3
SCHEMBL34462781 0.75 CLK4 (0.56) MAPTMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL19892519 0.74 L3MBTL1 (0.61) MAPTMEN1KMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117916237-A Amino aryl integrin agonist compounds 德克萨斯心脏研究所 2024-04-19 CN claimed
CN-117916237-A Amino aryl integrin agonist compounds 德克萨斯心脏研究所 2024-04-19 CN disclosed