SCHEMBL30858740

SCHEMBL30858740

N#Cc1cc(F)cc(N=C=O)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.35
CYP3A4 P08684 1/20 0.35
EPAS1 Q99814 2/20 0.33
GRM5 P41594 1/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21239456 1.00 TRPA1 (0.35) TRPA1CYP3A4EPAS1GRM5MAPK1
SCHEMBL159581 0.81 MAPK1 (0.41) TRPA1CYP3A4MAPK1TDP1
SCHEMBL19146345 0.81 MIF (0.34) GRM5
SCHEMBL8375351 0.80 EPAS1 (0.35) EPAS1GRM5
SCHEMBL1421650 0.73 GRM5 (0.47) GRM5
SCHEMBL56741 0.73 GRM5 (0.43) GRM5
SCHEMBL7921988 0.72 MAPK1 (0.44) TRPA1CYP3A4MAPK1TDP1
SCHEMBL4240933 0.72 CYP3A4 (0.41) TRPA1CYP3A4MAPK1TDP1
Isothiocyanate SCHEMBL3612486 0.72 MAPK1 (0.35) TRPA1CYP3A4MAPK1TDP1
SCHEMBL28560711 0.72 VCAM1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024067566-A1 SATURATED RING DERIVATIVE, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PHARMACEUTICAL USE THEREOF 苏州阿尔脉生物科技有限公司 2024-04-04 WO disclosed