Amisometradine

Amisometradine

SCHEMBL309300

C=C(C)Cn1c(N)cc(=O)n(C)c1=O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
CYP3A4 P08684 1/20 0.53
HPGD P15428 1/20 0.42
GAA P10253 2/20 0.39
L3MBTL1 Q9Y468 3/20 0.38
POLB P06746 1/20 0.36
HTT P42858 1/20 0.35
KDM4E B2RXH2 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
DPP4 P27487 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK1 P28482 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990525 0.80 ALDH1A1 (0.46) ALDH1A1CYP3A4HPGDGAAL3MBTL1
SCHEMBL17582653 0.77 ALDH1A1 (0.66) ALDH1A1CYP3A4HPGDGAAL3MBTL1
SCHEMBL6305749 0.75 ALDH1A1 (0.64) ALDH1A1CYP3A4HPGDGAAKDM4E
SCHEMBL19722541 0.74 HTT (0.43) ALDH1A1GAAPOLBHTTKDM4E
SCHEMBL22899026 0.74 HTT (0.47) ALDH1A1GAAPOLBHTTKDM4E
SCHEMBL4803924 0.73 ALDH1A1 (0.51) ALDH1A1CYP3A4HPGDGAAL3MBTL1
SCHEMBL10957985 0.72 ALDH1A1 (1.00) ALDH1A1CYP3A4HPGDGAAL3MBTL1
SCHEMBL22521705 0.71 HPGD (0.54) ALDH1A1CYP3A4HPGDGAAL3MBTL1
SCHEMBL4811069 0.71 MAPK1 (0.39) ALDH1A1HPGDPOLBHTTKDM4E
SCHEMBL9707792 0.70 ALDH1A1 (0.57) ALDH1A1CYP3A4HPGDPOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 541 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
EP-2560634-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS Piramal Enterprises Limited (IN) 2013-02-27 EP claimed
WO-2011132171-A1 NITRIC OXIDE RELEASING PRODRUGS OF THERAPEUTIC AGENTS PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-10-27 WO claimed
US-20110263526-A1 Nitric Oxide Releasing Prodrugs of Therapeutic Agents PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-10-27 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
WO-2006127024-A1 REAGENTS AND METHODS FOR LABELING TERMINAL OLEFINS EISAI CO. LTD. (JP) 2006-11-30 WO claimed
US-20060045846-A1 Reagents and methods for labeling terminal olefins EISAI R&D MANAGEMENT CO., LTD. (JP) 2006-03-02 US claimed
EP-1087953-B1 NITRATE SALTS OF ANTIHYPERTENSIVE MEDICINES NICOX SA (FR) 2004-11-17 EP claimed
CN-1315945-A Nitrate salts of antihypertensive drugs NICOX SA (FR) 2001-10-03 CN claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1087953-A1 NITRATE SALTS OF ANTIHYPERTENSIVE MEDICINES NICOX S.A. (FR) 2001-04-04 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-1999067231-A1 NITRATE SALTS OF ANTIHYPERTENSIVE MEDICINES NICOX S.A. (FR) 1999-12-29 WO claimed
US-4690824-A Solid pharmaceutical formulations for slow, zero order release via controlled surface erosion: expanded range REDI-ROWELL, INC. (US) 1987-09-01 US claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110263526-A1 Nitric Oxide Releasing Prodrugs of Therapeutic Agents NOS2, NOS1, NOS3 ALDH1A1 204/4885CYP3A4 68/4885HPGD 9/4885
US-20060045846-A1 Reagents and methods for labeling terminal olefins EEF2, RNF168, REL ALDH1A1 892/4885CYP3A4 426/4885HPGD 1653/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.