SCHEMBL3095656

SCHEMBL3095656

O=C(O)C1CCN(c2ccc(Cl)c(Cl)c2)C1=O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
SLC6A2 P23975 15/20 0.49
SLC6A4 P31645 15/20 0.49
SLC6A3 Q01959 12/20 0.49
PTPN1 P18031 1/20 0.46
CYP2D6 P10635 4/20 0.44
KCNH2 Q12809 4/20 0.44
ALDH1A1 P00352 1/20 0.42
ADAM17 P78536 1/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2289335 0.87 ALDH1A1 (0.46) NOTUMHDAC1HDAC8HDAC6PTPN1
SCHEMBL892162 0.87 PTPN1 (0.44) NOTUMHDAC1HDAC8HDAC6SLC6A2
SCHEMBL892180 0.83 PTPN1 (0.52) NOTUMHDAC1HDAC8HDAC6PTPN1
SCHEMBL892936 0.82 NOTUM (0.52) NOTUMHDAC1HDAC8HDAC6PTPN1
SCHEMBL7818940 0.81 SLC6A2 (0.54) NOTUMHDAC1HDAC8HDAC6SLC6A2
SCHEMBL7433338 0.80 HTT (0.52) NOTUMHDAC1HDAC8HDAC6SLC6A2
SCHEMBL893097 0.79 PTPN1 (0.46) PTPN1ALDH1A1CYP2C19
SCHEMBL892698 0.79 TSHR (0.55) NOTUMHDAC6PTPN1ALDH1A1
SCHEMBL308869 0.78 PTPN1 (0.59) NOTUMHDAC1HDAC8HDAC6PTPN1
SCHEMBL891655 0.77 TSHR (0.47) PTPN1CYP2D6ALDH1A1CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8324250-B2 Piperidine derivatives as NK3 receptor antagonists HOFFMANN-LA ROCHE INC. (US) 2012-12-04 US disclosed
US-20100256126-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE, INC. 2010-10-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100256126-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HTR3A, OPRL1, OPRK1 NOTUM 4676/4885HDAC1 1713/4885HDAC8 2297/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.