SCHEMBL30965201

SCHEMBL30965201

COc1ccc2[nH]nc(CC(=O)O)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
AKR1C2 P52895 2/20 0.56
PRKAG1 P54619 1/20 0.51
PRKAA1 Q13131 1/20 0.51
PRKAB1 Q9Y478 1/20 0.51
GSK3B P49841 4/20 0.47
HSD17B10 Q99714 3/20 0.47
PTGS1 P23219 2/20 0.47
AKR1C3 P42330 1/20 0.47
ALDH1A1 P00352 3/20 0.46
HPGD P15428 1/20 0.46
PTGS2 P35354 1/20 0.46
LMNA P02545 2/20 0.46
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 2/20 0.44
MAPT P10636 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14734878 0.83 KDM4E (0.50) KDM4EPRKAG1PRKAA1PRKAB1GSK3B
SCHEMBL27942416 0.82 PTGS2 (0.47) KDM4EGSK3BPTGS1PTGS2LMNA
SCHEMBL17232485 0.80 KDM4E (0.50) KDM4EPRKAG1PRKAA1PRKAB1HSD17B10
SCHEMBL5988579 0.80 TTK (0.53) KDM4EGSK3BHSD17B10ALDH1A1HPGD
SCHEMBL8151565 0.79 CNR2 (0.44) KDM4EAKR1C2PRKAG1PRKAA1PRKAB1
SCHEMBL17221269 0.79 HTR2B (0.53) KDM4EPRKAG1PRKAA1PRKAB1HSD17B10
SCHEMBL9295415 0.79 MTNR1A (0.52) KDM4EPRKAG1PRKAA1PRKAB1GSK3B
SCHEMBL7581326 0.78 LMNA (0.49) KDM4EPRKAG1PRKAA1PRKAB1GSK3B
SCHEMBL30965223 0.78 TSHR (0.54) KDM4EHSD17B10PTGS1ALDH1A1HPGD
SCHEMBL929332 0.78 PRKAG1 (0.79) KDM4EPRKAG1PRKAA1PRKAB1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024085695-A1 NOVEL ALTIRATINIB DERIVATIVE, MANUFACTURING METHOD THEREFOR, AND COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION, ALLEVIATION, OR TREATMENT OF SKIN PIGMENTATION 재단법인 아산사회복지재단 2024-04-25 WO disclosed