SCHEMBL30970488

SCHEMBL30970488

COc1c(C)c(-c2cc(C)ccc2S(=O)(=O)O)cc(-c2cc(C)ccc2S(=O)(=O)O)c1C(=O)N1Cc2ccc(N)cc2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.40
NR1H2 P55055 1/20 0.36
PDK2 Q15119 1/20 0.34
MMP8 P22894 4/20 0.34
MMP3 P08254 2/20 0.34
AVPR1B P47901 1/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA7 P43166 2/20 0.33
CA9 Q16790 2/20 0.33
CA14 Q9ULX7 2/20 0.33
DPP8 Q6V1X1 2/20 0.32
DPP9 Q86TI2 2/20 0.32
DPP7 Q9UHL4 1/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30970491 0.87 KCNA1 (0.36) HSP90AA1AVPR1BALDH1A1RECQLHPGD
SCHEMBL30970490 0.85 TRAP1 (0.33) HSP90AA1AVPR1BMEN1GAAKMT2A
SCHEMBL30368417 0.83 HSP90AA1 (0.44) HSP90AA1CA2ALDH1A1KDM4ETDP1
SCHEMBL30970484 0.80 TRAP1 (0.32) AVPR1BMEN1POLBGAAKMT2A
SCHEMBL30368050 0.76 HSP90AA1 (0.46) HSP90AA1CA2ALDH1A1KDM4ENAMPT
SCHEMBL30970485 0.74 HSP90AA1 (0.33) HSP90AA1ALDH1A1KDM4EMEN1GAA
SCHEMBL30970486 0.74 HSP90AA1 (0.33) HSP90AA1ALDH1A1KDM4EMEN1GAA
SCHEMBL30368298 0.74 HSP90AA1 (0.42) HSP90AA1CA2NAMPT
SCHEMBL31281629 0.73 NR1H2 (0.41) HSP90AA1NR1H2PDK2MMP8MMP3
SCHEMBL25214950 0.73 ALDH1A1 (0.39) HSP90AA1MMP8MMP3CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118317949-A Isoindolines as PMS2 inhibitors 奈奥芬莱有限公司 2024-07-09 CN disclosed