SCHEMBL309794

SCHEMBL309794

C1=Nc2ccccc2Nc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
GAA P10253 1/20 0.50
TRPA1 O75762 8/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
USP2 O75604 1/20 0.45
PPARG P37231 1/20 0.45
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
HSD17B10 Q99714 1/20 0.45
NR2E3 Q9Y5X4 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL2778281 0.85 MEN1 (0.39) MAPTGAATRPA1MEN1KMT2A
Maleic Acid SCHEMBL2778279 0.85 MEN1 (0.39) MAPTGAATRPA1MEN1KMT2A
SCHEMBL11499806 0.80 GAA (0.43) MAPTGAATRPA1MEN1KMT2A
SCHEMBL11162416 0.80 MEN1 (0.44) MAPTGAATRPA1MEN1KMT2A
SCHEMBL14128978 0.80 TRPA1 (0.44) MAPTGAATRPA1MEN1KMT2A
SCHEMBL7456203 0.80 TRPA1 (0.43) MAPTGAATRPA1MEN1KMT2A
SCHEMBL20067129 0.80 SMN1; SMN2 (0.43) MAPTGAATRPA1MEN1KMT2A
SCHEMBL8203995 0.80 BCHE (0.44) MAPTTRPA1MEN1KMT2AUSP2
SCHEMBL5138230 0.80 TRPA1 (0.47) MAPTGAATRPA1MEN1KMT2A
SCHEMBL20067134 0.80 ROS1 (0.42) MAPTGAATRPA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 228 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091050-A1 OLIGOMER-TRICYCLIC CONJUGATES NEKTAR THERAPEUTICS (US) 2011-07-28 WO claimed
JP-2011504928-A 2011-02-17 JP claimed
EP-2222342-A1 OLIGOMER-TRICYCLIC CONJUGATES Nektar Therapeutics (US) 2010-09-01 EP claimed
WO-2009073154-A1 OLIGOMER-TRICYCLIC CONJUGATES NEKTAR THERAPEUTICS AL, CORPORATION (US) 2009-06-11 WO claimed
US-6103715-A COMPOUNDS THAT BIND TO THE DOPAMINE D4 RECEPTOR AND THEIR USE AS ANXIOLYTIC AGENTS, TREATMENT FOR SCHIZOPHRENIA, AND DRUG SCREENING; SIDE EFFECT REDUCTIOON ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-15 US claimed
EP-0736024-A1 N-HETEROBICYCLYL-PIPERAZINYL OR-PIPERADINYL TRICYCLIC DERIVATIVES USEFUL AS DOPAMINE RECEPTOR LIGANDS Allelix Biopharmaceuticals Inc. (CA) 1996-10-09 EP claimed
US-5561127-A TREATING ANXIETY, SCHIZOPHRENIA ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1996-10-01 US claimed
WO-1996019479-A1 MUSCARINIC RECEPTOR LIGANDS ALLELIX BIOPHARMACEUTICALS INC. (US) 1996-06-27 WO claimed
WO-1995017400-A1 N-HETEROBICYCLYL-PIPERAZINYL OR-PIPERADINYL TRICYCLIC DERIVATIVES USEFUL AS DOPAMINE RECEPTOR LIGANDS ALLELIX BIOPHARMACEUTICALS INC. (CA) 1995-06-29 WO claimed
US-12403143-B2 Pharmaceutical composition for treating functional psychiatric disorders OBSCHESTVO S OGRANICHENNOI OTVETSTVENNOSTYU "VALENTEK" (RU) 2025-09-02 US disclosed
US-20250177354-A1 THERAPEUTIC COMBINATIONS, COMPOSITIONS, AND METHODS FOR DESIGNING AND PRODUCING ENTACTOGENIC MINDSTATES MINDSTATE DESIGN LABS INC (US) 2025-06-05 US disclosed
US-20250101104-A1 BISPECIFIC MOLECULE WITH TUNABLE AFFINITY TO A TARGETED ANTIGEN MABSWITCH INC (US) 2025-03-27 US disclosed
US-20250064992-A1 IMAGING METHOD FOR DESIGNER RECEPTOR, ANTAGONIST OR AGONIST, PHARMACEUTICAL, AND COMPANION DIAGNOSTIC AGENT NATIONAL INSTITUTES FOR QUANTUM AND RADIOLOGICAL SCIENCE AND TECHNOLOGY (JP) 2025-02-27 US disclosed
CN-119497589-A Therapeutic combinations, compositions and methods for designing and producing conditions that promote mental well-being 心境设计实验室股份有限公司 2025-02-21 CN disclosed
EP-0035714-A2 10-Substituted-5-cyanomethylene-10,11-dihydro-dibenzo-(a,d)-cycloheptenes, process for their preparation and pharmaceutical compositions containing them BASF Aktiengesellschaft (DE) 1981-09-16 EP disclosed
EP-0019172-A1 6-Substituted 11-alkylene-morphantridines, process for preparing them and pharmaceutical compositions containing them BASF Aktiengesellschaft (DE) 1980-11-26 EP disclosed
US-4191760-A ANTISCHIZOPHRENICS ABBOTT LABORATORIES (US) 1980-03-04 US disclosed
US-4096261-A ANTISCHIZOPHRENICS ABBOTT LABORATORIES (US) 1978-06-20 US disclosed
US-4054572-A Hexahydro pyridine [1,2d] dibenza [b,f] (1,4)-diazepines AKZONA INCORPORATED (US) 1977-10-18 US disclosed
US-3908010-A Basically substituted heterocycles as anti-emetics WANDER AG DR A 1975-09-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250064992-A1 IMAGING METHOD FOR DESIGNER RECEPTOR, ANTAGONIST OR AGONIST, PHARMACEUTICAL, AND COMPANION DIAGNOSTIC AGENT HTR3D, CHRNA4, CHRNA3 MAPT 1515/4885GAA 4485/4885TRPA1 646/4885
US-12403143-B2 Pharmaceutical composition for treating functional psychiatric disorders HTR5A, HTR2C, HTR2A MAPT 1179/4885GAA 3369/4885TRPA1 1158/4885
US-20250177354-A1 THERAPEUTIC COMBINATIONS, COMPOSITIONS, AND METHODS FOR DESIGNING AND PRODUCING ENTACTOGENIC MINDSTATES CNR2, CNR1, HTR6 MAPT 2221/4885GAA 4434/4885TRPA1 2986/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.