SCHEMBL30995146

SCHEMBL30995146

O=C(O)c1cc2c(F)cc(Br)cc2n1C1CCC1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.35
CYP11B2 P19099 2/20 0.34
MCL1 Q07820 1/20 0.33
PGR P06401 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HCAR3 P49019 1/20 0.32
NOTUM Q6P988 1/20 0.31
CCR2 P41597 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
DGAT1 O75907 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30995112 0.97 KDM5A (0.35) KDM5ACYP11B2MCL1PGRL3MBTL1
SCHEMBL30995171 0.94 CYP11B2 (0.38) KDM5ACYP11B2MCL1NOTUMCCR2
SCHEMBL30995137 0.83 WDR5 (0.36) MCL1L3MBTL1HCAR3CCR2
SCHEMBL30995240 0.81 ALDH1A1 (0.38) L3MBTL1MAPK1HTTKDM4EALDH1A1
SCHEMBL30995203 0.80 PKM (0.37) MAPK1HTTKDM4EALDH1A1HPGD
SCHEMBL30995195 0.80 NOTUM (0.42) CYP11B2MCL1L3MBTL1NOTUMALDH1A1
SCHEMBL30995218 0.79 ALDH1A1 (0.40) L3MBTL1MAPK1HTTKDM4EALDH1A1
SCHEMBL30995216 0.78 ADORA3 (0.32) PGR
SCHEMBL30995197 0.77 CYP11B2 (0.36) CYP11B2MCL1PGRL3MBTL1HCAR3
SCHEMBL30995185 0.76 MCL1 (0.46) MCL1L3MBTL1HCAR3CCR2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118530160-A Aromatic heterocyclic compound, preparation method and application thereof 上海翊石医药科技有限公司 2024-08-23 CN disclosed