SCHEMBL31146868

SCHEMBL31146868

O=C(Nc1cc2c(cc1I)OCO2)C(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.40
NPC1 O15118 5/20 0.39
RAB9A P51151 5/20 0.39
PKM P14618 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 8/20 0.38
MEN1 O00255 6/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 4/20 0.38
HPGD P15428 3/20 0.38
GAA P10253 1/20 0.38
KDM4E B2RXH2 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1744815 0.79 KDM4E (0.53) PTGS2NPC1RAB9AHSD17B10KMT2A
SCHEMBL19821774 0.69 ALDH1A1 (0.36) PTGS2NPC1RAB9AHSD17B10KMT2A
SCHEMBL31146876 0.67 GABRA1 (0.33) NPC1RAB9AHSD17B10TSHRKMT2A
SCHEMBL1742802 0.66 CYP3A4 (0.44) NPC1RAB9AHSD17B10KMT2AMEN1
SCHEMBL31709528 0.66 CYP3A4 (0.44) NPC1RAB9AHSD17B10KMT2AMEN1
SCHEMBL30015161 0.63 KDM4E (0.60) PKMHSD17B10TSHRKMT2AMEN1
SCHEMBL21721811 0.63 KDM4E (0.60) PKMHSD17B10TSHRKMT2AMEN1
SCHEMBL31146884 0.62 KDM4E (0.38) NPC1RAB9AKMT2AMEN1SMN1; SMN2
SCHEMBL31146894 0.61 CYP1A2 (0.40) NPC1RAB9AKMT2AMEN1SMN1; SMN2
SCHEMBL7813652 0.61 ALDH1A1 (0.46) PTGS2NPC1RAB9APKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4680606-A1 ADENINE DERIVATIVES AS HSP90 INHIBITORS AtmosR (FR) 2026-01-21 EP disclosed
WO-2024194175-A1 ADENINE DERIVATIVES AS HSP90 INHIBITORS ATMOSR (FR) 2024-09-26 WO disclosed